SCHEMBL9100034

SCHEMBL9100034

COc1cc(C(=O)N(NC(=O)c2ccc3c(c2C)OCCO3)C(C)(C)C)c(F)c(OC)c1C

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.43
GPX4 P36969 1/20 0.35
PLK1 P53350 1/20 0.34
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
TSHR P16473 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17424962 0.88 ABCB1 (0.42) ABCB1PLK1
SCHEMBL668808 0.86 ABCB1 (0.41) ABCB1NPC1MAPTRAB9A
SCHEMBL668714 0.85 ABCB1 (0.55) ABCB1PLK1
SCHEMBL668088 0.81 ABCB1 (0.53) ABCB1PLK1
SCHEMBL668264 0.81 ABCB1 (0.51) ABCB1PLK1
SCHEMBL5053915 0.78 ABCB1 (0.43) ABCB1SMN1; SMN2
SCHEMBL5057404 0.77 ABCB1 (0.57) ABCB1NPC1MAPTRAB9A
SCHEMBL667668 0.77 ABCB1 (0.39) ABCB1NPC1TSHRRAB9ASMN1; SMN2
SCHEMBL668764 0.77 ABCB1 (0.57) ABCB1
SCHEMBL5062349 0.77 CYP3A4 (0.46) ABCB1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2460786-A1 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex Intrexon Corporation (US) 2012-06-06 EP disclosed