SCHEMBL9102961

SCHEMBL9102961

CCc1c(OC)cccc1C(=O)N(NC(=O)c1cc(OC)c(OC)c(OC)c1)C(C)(C)C

nearest known ligand 0.68

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.53
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5053864 0.92 ABCB1 (0.61) ABCB1CYP3A4CYP2C9
SCHEMBL583844 0.89 ABCB1 (0.67) ABCB1CYP3A4
SCHEMBL8387173 0.86 ABCB1 (0.62) ABCB1
SCHEMBL5062581 0.84 ABCB1 (0.57) ABCB1CYP3A4CYP2C9
SCHEMBL17604610 0.83 ABCB1 (0.48) ABCB1
SCHEMBL5062538 0.83 ABCB1 (0.55) ABCB1
SCHEMBL5057173 0.83 ABCB1 (0.61) ABCB1CYP3A4CYP2C9
SCHEMBL9102034 0.82 ABCB1 (0.54) ABCB1
SCHEMBL18091869 0.81 ABCB1 (0.55) ABCB1
SCHEMBL64477 0.81 ABCB1 (0.77) ABCB1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2460786-B1 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex INTREXON CORP (US) 2016-01-13 EP disclosed
EP-2460786-A1 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex Intrexon Corporation (US) 2012-06-06 EP disclosed