SCHEMBL9103558

SCHEMBL9103558

CSc1ccc(Nc2c(OC(=O)NOCCO)cc3ccncn23)c(F)c1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.47
CYP2C9 P11712 2/20 0.45
MAP2K1 Q02750 14/20 0.38
MAP2K2 P36507 4/20 0.37
MAP2K5 Q13163 1/20 0.37
EIF2AK1 Q9BQI3 1/20 0.37
CYP2C19 P33261 1/20 0.36
ABCB11 O95342 1/20 0.35
NQO2 P16083 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9101063 0.89 MAP2K1 (0.43) KCNH2MAP2K1MAP2K2MAP2K5
SCHEMBL9104105 0.87 KCNH2 (0.62) KCNH2CYP2C9MAP2K1MAP2K2MAP2K5
SCHEMBL1977165 0.86 KCNH2 (0.59) KCNH2CYP2C9MAP2K1MAP2K2MAP2K5
SCHEMBL9885440 0.81 KCNH2 (0.53) KCNH2CYP2C9MAP2K1MAP2K2MAP2K5
SCHEMBL1615224 0.78 KCNH2 (0.76) KCNH2CYP2C9MAP2K1MAP2K2MAP2K5
SCHEMBL1976121 0.77 KCNH2 (0.47) KCNH2CYP2C9MAP2K1MAP2K2MAP2K5
SCHEMBL1977219 0.76 MAP2K2 (0.41) KCNH2CYP2C9MAP2K1MAP2K2CYP2C19
SCHEMBL1980901 0.76 MAP2K1 (0.43) KCNH2CYP2C9MAP2K1MAP2K2
SCHEMBL12646887 0.76 CYP2C9 (0.76) KCNH2CYP2C9MAP2K1MAP2K2MAP2K5
SCHEMBL9101056 0.76 MAP2K1 (0.53) KCNH2MAP2K1MAP2K2MAP2K5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2220092-B1 AZAINDOLIZINES AND METHODS OF USE GENENTECH INC (US) 2012-06-06 EP claimed