Hydrochlorthiazide

Hydrochlorthiazide

SCHEMBL9108846

COc1ccc2nc(C#N)sc2c1.c1cscn1

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2C19 P33261 2/20 0.47
PDK1 Q15118 1/20 0.46
MAPT P10636 6/20 0.45
RAB9A P51151 5/20 0.45
SMN1; SMN2 Q16637 5/20 0.45
NPC1 O15118 4/20 0.45
MEN1 O00255 4/20 0.45
KMT2A Q03164 4/20 0.45
HTT P42858 2/20 0.43
DYRK1A Q13627 1/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
APP P05067 4/20 0.43
GAA P10253 2/20 0.43
GLA P06280 1/20 0.43
ALDH1A1 P00352 1/20 0.43
CD274 Q9NZQ7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL906609 0.87 CYP1A2 (0.59) CYP1A2CYP3A4CYP2C19PDK1MAPT
Hydrochlorthiazide SCHEMBL9735331 0.82 CYP1A2 (0.51) CYP1A2CYP3A4CYP2C19PDK1MAPT
SCHEMBL26691830 0.79 NPC1 (0.51) CYP1A2CYP3A4CYP2C19PDK1MAPT
SCHEMBL5857526 0.76 NPC1 (0.54) CYP1A2CYP3A4CYP2C19PDK1RAB9A
SCHEMBL12336473 0.74 CYP3A4 (0.60) CYP1A2CYP3A4CYP2C19MAPTRAB9A
SCHEMBL8125517 0.74 APP (0.54) CYP1A2CYP3A4CYP2C19PDK1MAPT
SCHEMBL21412546 0.73 CYP1A2 (0.59) CYP1A2CYP3A4CYP2C19PDK1MAPT
SCHEMBL12312877 0.73 CYP3A4 (0.46) CYP1A2CYP3A4CYP2C19PDK1MAPT
SCHEMBL8773253 0.71 CA2 (0.46) CYP1A2CYP3A4CYP2C19PDK1MAPT
SCHEMBL492368 0.71 CYP3A4 (0.59) CYP3A4RAB9AKMT2AALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0527186-A4 UNIV ILLINOIS (US) 1995-01-18 EP disclosed
EP-0527186-A1 PHOTODYNAMIC PLANT DEFOLIANTS AND CHLOROPHYLL BIOSYNTHESIS MODULATORS The Board of Trustees for the University of Illinois (US) 1993-02-17 EP disclosed
WO-1991016820-A1 PHOTODYNAMIC PLANT DEFOLIANTS AND CHLOROPHYLL BIOSYNTHESIS MODULATORS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 1991-11-14 WO disclosed