SCHEMBL9109424

SCHEMBL9109424

CN1Cc2cc(-c3ccc(CC(C#N)NC(=O)C4(NC(=O)O)CCOCC4)cc3)ccc2S1(O)O

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSC P53634 20/20 0.52
CTSK P43235 5/20 0.52
KCNH2 Q12809 2/20 0.47
LTB4R Q15722 1/20 0.47
LTB4R2 Q9NPC1 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9109430 0.92 CTSC (0.54) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL2891013 0.88 CTSC (0.67) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL2888997 0.88 CTSC (0.67) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL2888989 0.88 CTSC (0.67) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL2887673 0.85 CTSC (0.49) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL2890780 0.83 CTSC (0.54) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL2890645 0.83 CTSC (0.68) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL9888342 0.82 CTSC (0.50) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL7876862 0.82 CTSC (0.50) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL2890779 0.81 CTSC (0.54) CTSCCTSKKCNH2LTB4RLTB4R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8193239-B2 Substituted 1-cyanoethylheterocyclylcarboxamide compounds ASTRAZENECA AB (SE) 2012-06-05 US disclosed