SCHEMBL9110149

SCHEMBL9110149

CC1Nc2ccncc2NC1=O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 3/20 0.59
BRPF1 P55201 1/20 0.59
GSK3B P49841 2/20 0.50
TSHR P16473 1/20 0.41
KDM4A O75164 1/20 0.39
KDM4B O94953 1/20 0.39
KDM5C P41229 1/20 0.39
KDM4C Q9H3R0 1/20 0.39
KDM5B Q9UGL1 1/20 0.39
KDM3A Q9Y4C1 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ADORA3 P0DMS8 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
XIAP P98170 1/20 0.35
BIRC2 Q13490 1/20 0.35
NTRK1 P04629 1/20 0.34
BRD4 O60885 4/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9110151 1.00 CREBBP (0.59) CREBBPBRPF1GSK3BTSHRKDM4A
SCHEMBL9414037 0.93 CREBBP (0.59) CREBBPBRPF1GSK3BTSHRKDM4A
Hydrochloric Acid SCHEMBL15953312 0.91 CREBBP (0.58) CREBBPBRPF1GSK3BTSHRKDM4A
SCHEMBL1101924 0.75 CREBBP (1.00) CREBBPBRPF1GSK3BTSHRMEN1
SCHEMBL10327064 0.75 CREBBP (1.00) CREBBPBRPF1GSK3BTSHRMEN1
SCHEMBL7668762 0.75 CREBBP (1.00) CREBBPBRPF1GSK3BTSHRMEN1
SCHEMBL13185757 0.73 PDE3B (0.43) CREBBPBRPF1GSK3BKDM4AKDM4B
SCHEMBL15314282 0.73 PDE3B (0.43) CREBBPBRPF1GSK3BKDM4AKDM4B
SCHEMBL25059407 0.72 ADORA3 (0.35) MEN1KMT2AADORA3ADORA2AADORA1
SCHEMBL9110204 0.70 GSK3B (0.45) CREBBPBRPF1GSK3BTSHRXIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5424311-A A viricides for treating viral diseases; HIV enzyme inhibitor HOESCHST AKTIENGESELLSCHAFT (DE) 1995-06-13 US disclosed
EP-0590428-A1 Azaquinoxalines, process for their preparation, and their use HOECHST AKTIENGESELLSCHAFT (DE) 1994-04-06 EP disclosed