SCHEMBL9114052

SCHEMBL9114052

COc1cc(CC(=O)NCC(c2ccccc2)c2ccccc2)cc(OC)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 3/20 0.64
L3MBTL1 Q9Y468 1/20 0.55
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
BCHE P06276 1/20 0.52
NPC1 O15118 1/20 0.51
MTNR1A P48039 2/20 0.50
MTNR1B P49286 2/20 0.50
CNR2 P34972 1/20 0.50
SIGMAR1 Q99720 1/20 0.49
ALDH1A1 P00352 2/20 0.49
GPR139 Q6DWJ6 1/20 0.49
LMNA P02545 1/20 0.48
ALPL P05186 1/20 0.48
MAPT P10636 1/20 0.48
ALOX12 P18054 1/20 0.48
HTT P42858 1/20 0.48
CNR1 P21554 1/20 0.48
CCR3 P51677 1/20 0.47
HDAC1 Q13547 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9114227 0.86 TACR1 (0.61) TACR1MEN1KMT2ABCHEMTNR1A
SCHEMBL9116017 0.86 MEN1 (0.68) TACR1L3MBTL1MEN1KMT2AMTNR1A
SCHEMBL9115325 0.80 MEN1 (0.75) TACR1MEN1KMT2ANPC1ALDH1A1
SCHEMBL8356709 0.79 TACR1 (0.55) TACR1MEN1KMT2ABCHELMNA
SCHEMBL9114494 0.74 TACR1 (0.64) TACR1L3MBTL1MEN1KMT2ASIGMAR1
SCHEMBL9117035 0.74 MTNR1A (0.65) TACR1MEN1KMT2AMTNR1AMTNR1B
SCHEMBL9468387 0.74 NPC1 (0.60) NPC1CNR2ALDH1A1MAPTHTT
SCHEMBL9113000 0.73 TACR1 (0.69) TACR1MEN1KMT2AMTNR1AMTNR1B
SCHEMBL30468424 0.72 CA1 (0.54) MTNR1AMTNR1BALDH1A1MAPTHTT
SCHEMBL228947 0.72 CA1 (0.54) MTNR1AMTNR1BALDH1A1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995011880-A1 SUBSTITUTED AMIDES AS TACHYKININ ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 1995-05-04 WO disclosed