SCHEMBL9114080

SCHEMBL9114080

CS(=O)(=O)Nc1ccc2c(c1)C(O)CC1(CCC(N3CCc4ccccc4C3)CC1)O2

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.59
HTR1A P08908 1/20 0.37
HTR7 P34969 1/20 0.37
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
PRMT5 O14744 2/20 0.36
TRPV1 Q8NER1 1/20 0.36
WDR77 Q9BQA1 1/20 0.35
ADRA1D P25100 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9115512 0.88 KCNH2 (0.76) KCNH2
SCHEMBL9112284 0.88 KCNH2 (0.47) KCNH2HDAC3HDAC4HDAC1HDAC7
SCHEMBL9113519 0.86 HRH3 (0.44) KCNH2HTR1AHTR7
Hydrochloric Acid SCHEMBL8831795 0.84 KCNH2 (0.78) KCNH2HTR1AHTR7HDAC3HDAC4
Hydrochloric Acid SCHEMBL8831789 0.84 KCNH2 (0.78) KCNH2HTR1AHTR7HDAC3HDAC4
SCHEMBL9115697 0.82 ADRA1D (0.53) KCNH2ADRA1D
Hydrochloric Acid SCHEMBL8832001 0.79 KCNH2 (0.83) KCNH2
SCHEMBL9114263 0.78 KCNH2 (0.38) KCNH2HTR1AHTR7PRMT5WDR77
SCHEMBL9115004 0.78 KCNH2 (0.40) KCNH2HTR1AHTR7
Hydrochloric Acid SCHEMBL8832008 0.76 KCNH2 (0.79) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995014469-A1 NOVEL SPIROCYCLES MERCK & CO., INC. (US) 1995-06-01 WO disclosed
US-5403846-A Antiarrhythmic agents MERCK & CO., INC. (US) 1995-04-04 US disclosed