SCHEMBL9116533

SCHEMBL9116533

COc1cc(O)c(C(=O)CCCCBr)c(OC)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.59
CYP2D6 P10635 2/20 0.59
CYP2C19 P33261 1/20 0.59
USP2 O75604 1/20 0.56
MAPK1 P28482 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
LMNA P02545 1/20 0.51
HTR1A P08908 1/20 0.51
ADRA2A P08913 1/20 0.51
ADRA2C P18825 1/20 0.51
OPRK1 P41145 1/20 0.51
KCNH2 Q12809 1/20 0.51
EBP Q15125 1/20 0.51
SIGMAR1 Q99720 1/20 0.51
HRH3 Q9Y5N1 1/20 0.51
NFKB1 P19838 2/20 0.50
NFKB2 Q00653 2/20 0.50
RELA Q04206 2/20 0.50
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9117522 0.99 CYP3A4 (0.58) CYP3A4CYP2D6CYP2C19USP2MAPK1
SCHEMBL30506420 0.87 MEN1 (0.63) CYP3A4CYP2D6CYP2C19USP2MAPK1
SCHEMBL25304726 0.85 CYP3A4 (0.59) CYP3A4CYP2D6CYP2C19USP2MAPK1
SCHEMBL7192880 0.82 CYP3A4 (0.63) CYP3A4CYP2D6CYP2C19USP2MAPK1
SCHEMBL30506419 0.79 CYP3A4 (0.67) CYP3A4CYP2D6CYP2C19USP2MAPK1
SCHEMBL21275479 0.79 CYP3A4 (0.67) CYP3A4CYP2D6CYP2C19USP2MAPK1
SCHEMBL30002388 0.79 CYP3A4 (0.67) CYP3A4CYP2D6CYP2C19USP2MAPK1
SCHEMBL2874467 0.79 CYP3A4 (0.67) CYP3A4CYP2D6CYP2C19USP2MAPK1
SCHEMBL7901522 0.77 CYP3A4 (0.65) CYP3A4CYP2D6CYP2C19USP2MAPK1
SCHEMBL13002149 0.77 FFAR1 (0.63) CYP3A4NFKB1NFKB2RELAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995025731-A1 NOVEL 3-(φ-(4-BENZOYLPIPERIDINO)ALKYL)-4H-BENZOPYRAN-4-ONES, PREPARATION AND THERAPEUTICAL USE THEREOF PIERRE FABRE MEDICAMENT (FR) 1995-09-28 WO disclosed