SCHEMBL9116772

SCHEMBL9116772

Cc1ccc(C2=CC3(C=C2c2ccc(S(N)(=O)=O)cc2)CCC3)cn1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.51
PTGS1 P23219 6/20 0.47
CA2 P00918 9/20 0.41
CA9 Q16790 9/20 0.41
CA1 P00915 7/20 0.41
CA12 O43570 7/20 0.41
CA5A P35218 3/20 0.41
CA5B Q9Y2D0 3/20 0.41
CA4 P22748 2/20 0.41
ALOX5AP P20292 1/20 0.36
CA3 P07451 1/20 0.36
CA6 P23280 1/20 0.36
CA7 P43166 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9118146 0.97 PTGS2 (0.51) PTGS2PTGS1CA2CA9CA1
SCHEMBL9117172 0.95 PTGS2 (0.53) PTGS2PTGS1CA2CA9CA1
SCHEMBL9117471 0.88 PTGS2 (0.57) PTGS2PTGS1ALOX5AP
SCHEMBL9119469 0.86 PTGS2 (0.57) PTGS2PTGS1
SCHEMBL9115408 0.85 PTGS2 (0.47) PTGS2PTGS1CA2CA9CA1
SCHEMBL9117574 0.85 PTGS2 (0.46) PTGS2PTGS1CA2CA9CA1
SCHEMBL9116743 0.84 PTGS2 (0.40) PTGS2PTGS1CA2CA9CA1
SCHEMBL9118531 0.84 CA1 (0.55) PTGS2PTGS1CA2CA9CA1
SCHEMBL9117882 0.84 CA12 (0.55) PTGS2PTGS1CA2CA9CA1
SCHEMBL9117164 0.84 PTGS2 (0.42) PTGS2PTGS1CA2CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030652-A1 SUBSTITUTED SPIRODIENES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO claimed
WO-1995030652-A1 SUBSTITUTED SPIRODIENES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed