SCHEMBL9117259

SCHEMBL9117259

O=C1[C@H]2CCC[C@H]2N(C(=O)CCCCBr)c2ccccc2N1Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.47
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
POLB P06746 1/20 0.47
MT-CO2 P00403 1/20 0.39
ALOX5 P09917 1/20 0.39
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
CRHBP P24387 1/20 0.38
CRHR2 Q13324 1/20 0.38
KCNH2 Q12809 1/20 0.38
XIAP P98170 4/20 0.37
CYP3A4 P08684 2/20 0.37
MAPK1 P28482 1/20 0.37
BRD4 O60885 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9117256 1.00 ALDH1A1 (0.47) ALDH1A1KMT2AMEN1POLBMT-CO2
SCHEMBL9115888 0.99 ALDH1A1 (0.46) ALDH1A1KMT2AMEN1POLBMT-CO2
SCHEMBL9118170 0.89 ALDH1A1 (0.49) ALDH1A1KMT2AMEN1POLBMT-CO2
SCHEMBL9118163 0.89 ALDH1A1 (0.49) ALDH1A1KMT2AMEN1POLBMT-CO2
SCHEMBL7495825 0.88 ALDH1A1 (0.52) ALDH1A1KMT2AMEN1POLBMT-CO2
SCHEMBL7500262 0.88 ALDH1A1 (0.52) ALDH1A1KMT2AMEN1POLBMT-CO2
SCHEMBL7501691 0.86 SMN1; SMN2 (0.48) ALDH1A1KMT2AMEN1POLBMAPK1
SCHEMBL7497359 0.85 ALDH1A1 (0.53) ALDH1A1KMT2AMEN1POLBMT-CO2
SCHEMBL7497354 0.85 ALDH1A1 (0.53) ALDH1A1KMT2AMEN1POLBMT-CO2
SCHEMBL7498239 0.84 ALDH1A1 (0.52) ALDH1A1KMT2AMEN1POLBMT-CO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995029900-A1 CONDENSED HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE AS GnRH ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-11-09 WO disclosed