SCHEMBL9117464

SCHEMBL9117464

Cc1ccc(C2=CC3(C=C2c2ccc(S(N)(=O)=O)cc2)CCC3)nc1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.51
PTGS1 P23219 4/20 0.40
CA2 P00918 7/20 0.40
CA1 P00915 6/20 0.40
CA9 Q16790 6/20 0.40
CA5A P35218 5/20 0.40
CA5B Q9Y2D0 5/20 0.40
CA12 O43570 3/20 0.40
CA3 P07451 1/20 0.40
CA6 P23280 1/20 0.40
CA7 P43166 1/20 0.40
CA4 P22748 3/20 0.39
ALOX5AP P20292 1/20 0.38
GRIA2 P42262 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9117163 0.98 PTGS2 (0.51) PTGS2PTGS1CA2CA1CA9
SCHEMBL9118062 0.95 PTGS2 (0.53) PTGS2PTGS1CA2CA1CA9
SCHEMBL9116432 0.93 PTGS2 (0.43) PTGS2PTGS1CA2CA1CA9
SCHEMBL9239184 0.91 PTGS2 (0.43) PTGS2PTGS1CA2CA1CA9
SCHEMBL9118699 0.89 PTGS2 (0.53) PTGS2PTGS1ALOX5APGRIA2
SCHEMBL9117725 0.88 PTGS2 (0.45) PTGS2PTGS1CA2CA1CA9
SCHEMBL9117472 0.87 PTGS2 (0.53) PTGS2PTGS1ALOX5APGRIA2
SCHEMBL9117882 0.86 CA12 (0.55) PTGS2PTGS1CA2CA1CA9
SCHEMBL9118587 0.86 PTGS2 (0.43) PTGS2PTGS1CA2CA1CA9
SCHEMBL9116766 0.86 PTGS2 (0.49) PTGS2PTGS1CA2CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030652-A1 SUBSTITUTED SPIRODIENES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO claimed
WO-1995030652-A1 SUBSTITUTED SPIRODIENES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed