SCHEMBL9119157

SCHEMBL9119157

COC(=O)CCCOc1ccc(CCC(=O)OC)c(OCCCCCO)c1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.52
ALDH1A1 P00352 1/20 0.52
KMT2A Q03164 1/20 0.52
MAPT P10636 1/20 0.45
CNR2 P34972 10/20 0.44
CNR1 P21554 6/20 0.44
PDE3B Q13370 3/20 0.43
PDE3A Q14432 3/20 0.43
P2RY12 Q9H244 3/20 0.43
PPARD Q03181 1/20 0.43
LTB4R Q15722 1/20 0.43
LTB4R2 Q9NPC1 1/20 0.43
TSHR P16473 1/20 0.43
PPARG P37231 1/20 0.42
PPARA Q07869 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9121261 0.88 PDE3B (0.46) MEN1ALDH1A1KMT2AMAPTCNR2
SCHEMBL27088423 0.88 MEN1 (0.67) MEN1ALDH1A1KMT2ACNR2CNR1
SCHEMBL9120001 0.86 MEN1 (0.47) MEN1ALDH1A1KMT2AMAPTCNR2
SCHEMBL9444512 0.86 CNR2 (0.43) MEN1ALDH1A1KMT2AMAPTCNR2
SCHEMBL8799495 0.86 MEN1 (0.48) MEN1ALDH1A1KMT2AMAPTCNR2
SCHEMBL9122500 0.81 PPARD (0.53) ALDH1A1PPARDLTB4RLTB4R2PPARG
SCHEMBL31155834 0.80 MEN1 (0.48) MEN1ALDH1A1KMT2AMAPTCNR2
SCHEMBL5988709 0.80 KMT2A (0.44) MEN1ALDH1A1KMT2AMAPTCNR2
SCHEMBL9120954 0.79 BRD4 (0.48) MEN1KMT2ACNR2PDE3BPDE3A
SCHEMBL9121657 0.78 HDAC8 (0.53) MAPTPDE3BPDE3AP2RY12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5434186-A Antiinflammatory agents HOFFMANN-LA ROCHE INC. (US) 1995-07-18 US disclosed
US-5273999-A A 4-keto-boroalkyleneoxychroman or 2,3-dihydrobenzofuran derivative HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed
EP-0531823-A1 Bicyclic carboxylic acid derivatives as anti-inflammatory agents F. HOFFMANN-LA ROCHE AG (CH) 1993-03-17 EP disclosed