SCHEMBL9119331

SCHEMBL9119331

COC(=O)c1cc(C)cnc1Br

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.47
OPRK1 P41145 5/20 0.45
CYP46A1 Q9Y6A2 1/20 0.43
KDM4E B2RXH2 4/20 0.40
GLA P06280 2/20 0.40
MAPK1 P28482 1/20 0.40
LMNA P02545 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TSHR P16473 2/20 0.39
HTT P42858 1/20 0.38
ABL1 P00519 1/20 0.38
ALDH1A1 P00352 2/20 0.38
SORT1 Q99523 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MAPT P10636 1/20 0.38
GAA P10253 1/20 0.38
NR4A2 P43354 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20872624 0.84 OPRK1 (0.51) OPRK1KDM4EMAPK1LMNASMN1; SMN2
SCHEMBL3108102 0.83 TSHR (0.46) KDM4EGLAMAPK1SMN1; SMN2TSHR
SCHEMBL12024798 0.81 ATM (0.50) ATMOPRK1CYP46A1KDM4EGLA
SCHEMBL30294812 0.81 OPRK1 (0.46) OPRK1KDM4EGLAMAPK1LMNA
SCHEMBL22288713 0.81 OPRK1 (0.46) ATMOPRK1KDM4EGLAMAPK1
SCHEMBL28956660 0.81 KDM4E (0.45) OPRK1KDM4EGLAMAPK1LMNA
SCHEMBL28960417 0.81 OPRK1 (0.46) OPRK1KDM4EGLAMAPK1LMNA
SCHEMBL19682934 0.81 KDR (0.49) OPRK1KDM4EMAPK1LMNAHTT
SCHEMBL29833413 0.80 ATM (0.49) ATMOPRK1CYP46A1KDM4EGLA
SCHEMBL2487068 0.80 ATM (0.49) ATMOPRK1CYP46A1KDM4EGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023218023-A1 THIAZOLOARYL-METHYL SUBSTITUTED CYCLIC HYDRAZINE-N-CARBOXAMIDE DERIVATIVES IDORSIA PHARMACEUTICALS LTD (CH) 2023-11-16 WO disclosed
US-5426089-A Controlling undesired plant growth SHELL RESEARCH LIMITED (GB) 1995-06-20 US disclosed
EP-0434132-B1 Herbicidal acrylonitrile derivatives SHELL INT RESEARCH (NL) 1995-04-05 EP disclosed
US-5366956-A Herbicidal acrylonitrile derivatives SHELL RESEARCH LIMITED (GB) 1994-11-22 US disclosed
EP-0434132-A2 Herbicidal acrylonitrile derivatives SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1991-06-26 EP disclosed