SCHEMBL9119490

SCHEMBL9119490

C[C@H]([C@](O)(Cn1cncn1)c1ccc(F)cc1F)S(=O)(=O)N1CCN(c2ccc(-n3cnn(CC(F)(F)F)c3=O)cc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 17/20 0.47
CYP2C9 P11712 13/20 0.47
CYP2C19 P33261 12/20 0.47
LMNA P02545 2/20 0.47
CYP2B6 P20813 1/20 0.47
CYP3A5 P20815 1/20 0.47
CYP3A7 P24462 1/20 0.47
MAPK1 P28482 1/20 0.47
CYP3A43 Q9HB55 1/20 0.47
CYP46A1 Q9Y6A2 1/20 0.47
CYP1A2 P05177 7/20 0.43
CYP2D6 P10635 7/20 0.43
KCNH2 Q12809 3/20 0.43
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9119798 0.89 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19LMNACYP2B6
SCHEMBL6942811 0.88 CYP3A4 (0.49) CYP3A4CYP2C9CYP2C19LMNACYP2B6
SCHEMBL9121596 0.88 CYP3A4 (0.52) CYP3A4CYP2C9CYP2C19LMNACYP2B6
SCHEMBL9121838 0.88 LMNA (0.48) CYP3A4CYP2C9CYP2C19LMNACYP2B6
SCHEMBL9119955 0.87 CYP3A4 (0.46) CYP3A4CYP2C9CYP2C19LMNACYP2B6
SCHEMBL9122049 0.85 CYP3A4 (0.51) CYP3A4CYP2C9CYP2C19LMNACYP2B6
SCHEMBL9121500 0.84 CYP3A4 (0.51) CYP3A4CYP2C9CYP2C19LMNACYP2B6
SCHEMBL6943875 0.82 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19LMNACYP2B6
SCHEMBL9119030 0.81 CYP3A4 (0.60) CYP3A4CYP2C9CYP2C19LMNACYP2B6
SCHEMBL9122301 0.81 CYP3A4 (0.58) CYP3A4CYP2C9CYP2C19LMNACYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5389663-A Fungicides TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-02-14 US disclosed
EP-0510700-A2 Azole compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-10-28 EP disclosed