SCHEMBL9120397

SCHEMBL9120397

CCC(C)n1ncn(-c2ccc(N3CCN(S[C@H](C)[C@](O)(Cn4cncn4)c4ccc(F)cc4F)CC3)cc2)c1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.49
LMNA P02545 3/20 0.49
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
GAA P10253 1/20 0.49
HTT P42858 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CYP3A4 P08684 17/20 0.47
CYP2C9 P11712 8/20 0.47
CYP2C19 P33261 7/20 0.47
CYP1A2 P05177 5/20 0.46
CYP2D6 P10635 5/20 0.46
MAPK1 P28482 2/20 0.46
CYP2B6 P20813 1/20 0.46
CYP3A5 P20815 1/20 0.46
CYP3A7 P24462 1/20 0.46
CYP3A43 Q9HB55 1/20 0.46
CYP46A1 Q9Y6A2 1/20 0.46
ABCB11 O95342 2/20 0.46
ABCG2 Q9UNQ0 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6938477 0.90 LMNA (0.51) MAPTLMNAKDM4EALDH1A1GAA
SCHEMBL9119955 0.88 CYP3A4 (0.46) LMNACYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL9121838 0.87 LMNA (0.48) MAPTLMNAKDM4EALDH1A1GAA
SCHEMBL9120402 0.87 HDAC3 (0.47) LMNACYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL9121521 0.84 CYP3A4 (0.54) LMNACYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL6938539 0.84 CYP3A4 (0.50) MAPTLMNAKDM4EALDH1A1GAA
SCHEMBL6942294 0.84 CYP3A4 (0.50) MAPTLMNAKDM4EALDH1A1GAA
SCHEMBL6936623 0.84 CYP3A4 (0.50) MAPTLMNAKDM4EALDH1A1GAA
SCHEMBL6944059 0.84 CYP3A4 (0.50) MAPTLMNAKDM4EALDH1A1GAA
SCHEMBL6940912 0.84 CYP3A4 (0.51) MAPTLMNAKDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5389663-A Fungicides TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-02-14 US disclosed
EP-0510700-A2 Azole compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-10-28 EP disclosed