SCHEMBL9124668

SCHEMBL9124668

CN(CCOc1ccc(/C=C2\SC(=O)NC2=O)cc1)C(=O)CCc1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HPGD P15428 9/20 0.68
PTPN1 P18031 2/20 0.58
MAOA P21397 2/20 0.58
MAOB P27338 2/20 0.58
POLB P06746 1/20 0.58
PPARG P37231 4/20 0.57
PIM1 P11309 2/20 0.55
PIM2 Q9P1W9 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9124675 1.00 HPGD (0.68) HPGDPTPN1MAOAMAOBPOLB
SCHEMBL9123327 0.90 HPGD (0.64) HPGDPTPN1MAOAMAOBPOLB
SCHEMBL9121091 0.90 HPGD (0.64) HPGDPTPN1MAOAMAOBPOLB
SCHEMBL9124681 0.89 HPGD (0.53) HPGDPTPN1MAOAMAOBPOLB
SCHEMBL9536304 0.84 HPGD (0.64) HPGDPTPN1MAOAMAOBPOLB
SCHEMBL9536301 0.84 HPGD (0.64) HPGDPTPN1MAOAMAOBPOLB
SCHEMBL8458670 0.84 PPARG (0.61) HPGDPTPN1MAOAMAOBPOLB
SCHEMBL8458668 0.84 PPARG (0.61) HPGDPTPN1MAOAMAOBPOLB
SCHEMBL6969911 0.83 HPGD (0.78) HPGDPTPN1MAOAMAOBPOLB
SCHEMBL6969914 0.83 HPGD (0.78) HPGDPTPN1MAOAMAOBPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5478851-A Hyperglycemic agent and antilipemic agent BEECHAM GROUP PLC (GB) 1995-12-26 US claimed
US-5478851-A Hyperglycemic agent and antilipemic agent BEECHAM GROUP PLC (GB) 1995-12-26 US disclosed
EP-0555264-A1 NOVEL COMPOUNDS BEECHAM GROUP plc (GB) 1993-08-18 EP disclosed
WO-1992007850-A1 NOVEL COMPOUNDS BEECHAM GROUP PLC (GB) 1992-05-14 WO disclosed