SCHEMBL9125331

SCHEMBL9125331

COC(=O)c1cccc2cc(Cl)ccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 2/20 0.54
ABL1 P00519 1/20 0.53
SLC6A4 P31645 2/20 0.50
SLC6A3 Q01959 2/20 0.50
RXFP1 Q9HBX9 1/20 0.49
CHEK1 O14757 1/20 0.48
KDM4E B2RXH2 2/20 0.48
NPSR1 Q6W5P4 2/20 0.48
ALDH1A1 P00352 1/20 0.48
HPGD P15428 1/20 0.48
PDE4B Q07343 1/20 0.47
SCN9A Q15858 1/20 0.47
PLA2G2A P14555 2/20 0.46
MEN1 O00255 2/20 0.46
MAPT P10636 2/20 0.46
KMT2A Q03164 2/20 0.46
LMNA P02545 2/20 0.46
HTT P42858 1/20 0.46
RAB9A P51151 1/20 0.45
SLC6A2 P23975 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29374722 1.00 NR4A2 (0.54) NR4A2ABL1SLC6A4SLC6A3RXFP1
SCHEMBL3571702 0.87 NR4A2 (0.54) NR4A2ABL1SLC6A4SLC6A3RXFP1
SCHEMBL29792644 0.87 NR4A2 (0.54) NR4A2ABL1SLC6A4SLC6A3RXFP1
SCHEMBL4961105 0.87 PTPN1 (0.45) NR4A2KDM4EALDH1A1HPGDMEN1
SCHEMBL19733167 0.83 ALDH1A1 (0.56) SLC6A4SLC6A3KDM4ENPSR1ALDH1A1
SCHEMBL13576763 0.82 KDM4E (0.60) NR4A2ABL1SLC6A4SLC6A3KDM4E
SCHEMBL30571222 0.82 CA12 (0.54) SLC6A4SLC6A3KDM4ENPSR1ALDH1A1
SCHEMBL69179 0.82 LCK (0.58) SLC6A4SLC6A3KDM4ENPSR1ALDH1A1
SCHEMBL343944 0.82 NR4A2 (0.53) NR4A2SLC6A4SLC6A3KDM4ENPSR1
SCHEMBL30213808 0.82 LCK (0.58) SLC6A4SLC6A3KDM4ENPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5395849-A Hybrid antitumor compounds containing a cyclic enediyne and a DNA-binder BRISTOL-MYERS SQUIBB COMPANY (US) 1995-03-07 US disclosed