SCHEMBL9127331

SCHEMBL9127331

CC1CC2=C(CSc3ccccc3)C(=O)CC[C@]2(C)[C@@H]2CC[C@@]3(C)[C@@H](CCC3(C)O)[C@H]12

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SHBG P04278 5/20 0.53
ALDH1A1 P00352 2/20 0.43
CYP19A1 P11511 9/20 0.41
AR P10275 4/20 0.40
NR3C1 P04150 1/20 0.36
PGR P06401 1/20 0.36
ADRA1A P35348 1/20 0.36
HTR2B P41595 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9127322 1.00 SHBG (0.53) SHBGALDH1A1CYP19A1ARNR3C1
SCHEMBL11522845 0.85 CYP19A1 (0.51) SHBGALDH1A1CYP19A1NR3C1PGR
SCHEMBL11522842 0.85 CYP19A1 (0.51) SHBGALDH1A1CYP19A1NR3C1PGR
SCHEMBL9124485 0.79 SHBG (0.41) SHBGALDH1A1CYP19A1ARNR3C1
SCHEMBL9124492 0.79 SHBG (0.41) SHBGALDH1A1CYP19A1ARNR3C1
SCHEMBL9125973 0.76 SHBG (0.63) SHBGALDH1A1CYP19A1ARNR3C1
SCHEMBL9125965 0.76 SHBG (0.63) SHBGALDH1A1CYP19A1ARNR3C1
SCHEMBL9541910 0.75 CYP19A1 (0.40) SHBGALDH1A1CYP19A1NR3C1PGR
SCHEMBL9541172 0.75 CYP19A1 (0.40) SHBGALDH1A1CYP19A1NR3C1PGR
SCHEMBL9541167 0.75 CYP19A1 (0.40) SHBGALDH1A1CYP19A1NR3C1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5389624-A Antiandrogenic [3,2-c]pyrazole and [3,2-d]triazole steroids SCHERING AKTIENGESELLSCHAFT (DE) 1995-02-14 US disclosed
US-5236912-A Treating prostate hyperplasia and carcinoma SCHERING AKTIENGESELLSCHAFT (DE) 1993-08-17 US disclosed
WO-1993013122-A1 3-METHYLSULPHONYLHYDRAZONO AND 3-OXYIMINO STEROIDS, A METHOD OF PREPARING THEM, PHARMACEUTICAL PREPARATIONS CONTAINING THEM AND THEIR USE IN THE PREPARATION OF DRUGS SCHERING AKTIENGESELLSCHAFT (DE) 1993-07-08 WO disclosed