SCHEMBL9130686

SCHEMBL9130686

CN(C)c1ccc(C(=O)C#Cc2ccncc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
APP P05067 4/20 0.68
VCP P55072 1/20 0.47
MAPT P10636 4/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
KDM4E B2RXH2 1/20 0.46
GFER P55789 1/20 0.46
CHRM5 P08912 1/20 0.46
CHKA P35790 1/20 0.46
RAB9A P51151 4/20 0.45
NPC1 O15118 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
MEN1 O00255 1/20 0.45
ALOX15 P16050 1/20 0.45
CASP1 P29466 1/20 0.45
HBB P68871 1/20 0.45
KMT2A Q03164 1/20 0.45
MPO P05164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9073927 0.94 APP (0.68) APPVCPMAPTALDH1A1HPGD
SCHEMBL9131883 0.84 APP (0.59) APPVCPMAPTALDH1A1HPGD
SCHEMBL9132523 0.84 APP (0.49) APPVCPMAPTALDH1A1GFER
SCHEMBL9184573 0.80 APP (0.51) APPMAPTALDH1A1HPGDKDM4E
SCHEMBL28972857 0.79 APP (0.69) APPVCPMAPTALDH1A1HPGD
SCHEMBL9069649 0.78 VCP (0.59) APPVCPMAPTALDH1A1HPGD
SCHEMBL9131641 0.78 APP (0.56) APPVCPMAPTALDH1A1HPGD
SCHEMBL9804473 0.77 CHRM5 (0.62) APPMAPTALDH1A1CHRM5CHKA
SCHEMBL9131344 0.77 APP (0.62) APPVCPMAPTALDH1A1HPGD
SCHEMBL9131411 0.76 APP (0.61) APPVCPMAPTALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0476658-B1 1-Phenyl-3-phenyl-2-propyne-1-ones MERRELL DOW PHARMA (US) 1995-11-15 EP claimed
EP-0476645-B1 Calcium uptake inhibitors MERRELL DOW PHARMA (US) 1995-09-06 EP claimed
US-5223518-A Controlling intake in leukocytes and platelets MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-29 US claimed
EP-0476645-A1 Calcium uptake inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1992-03-25 EP claimed
EP-0476658-B1 1-Phenyl-3-phenyl-2-propyne-1-ones MERRELL DOW PHARMA (US) 1995-11-15 EP disclosed
EP-0476645-B1 Calcium uptake inhibitors MERRELL DOW PHARMA (US) 1995-09-06 EP disclosed
US-5446068-A Antiinflammatory agent MERRELL DOW PHARMACEUTICALS INC. (US) 1995-08-29 US disclosed
US-5409942-A Administering 1-phenyl-3-aryl-2-propyne-1-ones compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1995-04-25 US disclosed
US-5248825-A Aromatic ketones containing triple bond MERRELL DOW PHARMACEUTICALS INC. (US) 1993-09-28 US disclosed
US-5223518-A Controlling intake in leukocytes and platelets MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-29 US disclosed
EP-0476645-A1 Calcium uptake inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1992-03-25 EP disclosed
EP-0476658-A1 1-Phenyl-3-phenyl-2-propyne-1-ones MERRELL DOW PHARMACEUTICALS INC. (US) 1992-03-25 EP disclosed