SCHEMBL9130944

SCHEMBL9130944

C#CC(O)c1ccc(N(CC)CC)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.49
TSHR P16473 2/20 0.49
CNR2 P34972 10/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
PSMD14 O00487 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPK1 P28482 1/20 0.44
RECQL P46063 1/20 0.44
GFER P55789 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
ALDH3A1 P30838 1/20 0.41
ALDH1A3 P47895 1/20 0.41
KDM4E B2RXH2 1/20 0.41
GAA P10253 1/20 0.41
GRK6 P43250 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 1/20 0.39
HSP90AA1 P07900 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6971747 0.79 ALDH1A1 (0.46) ALDH1A1TSHRL3MBTL1CYP3A4MAPK1
SCHEMBL4116469 0.78 ALDH1A1 (0.56) ALDH1A1TSHRCNR2L3MBTL1PSMD14
SCHEMBL29184903 0.77 ESR1 (0.46) TSHR
SCHEMBL9158083 0.76 ALDH1A1 (0.55) ALDH1A1TSHRCNR2L3MBTL1PSMD14
SCHEMBL9133521 0.76 ALDH1A1 (0.44) ALDH1A1TSHRCNR2L3MBTL1PSMD14
SCHEMBL4050620 0.75 CNR2 (0.47) ALDH1A1TSHRCNR2L3MBTL1PSMD14
SCHEMBL7201693 0.75 TSHR (0.45) ALDH1A1TSHRL3MBTL1MAPK1TDP1
SCHEMBL11433950 0.74 ALDH1A1 (0.58) ALDH1A1TSHRCNR2L3MBTL1PSMD14
SCHEMBL9131897 0.74 ALDH1A1 (0.42) ALDH1A1TSHRCNR2L3MBTL1PSMD14
SCHEMBL131813 0.73 ALDH1A1 (0.56) ALDH1A1TSHRCNR2L3MBTL1PSMD14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0476645-B1 Calcium uptake inhibitors MERRELL DOW PHARMA (US) 1995-09-06 EP disclosed
US-5409942-A Administering 1-phenyl-3-aryl-2-propyne-1-ones compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1995-04-25 US disclosed
EP-0250193-B1 Photoreactive lenses MARCONI GEC LTD (GB) 1993-10-27 EP disclosed
US-5223518-A Controlling intake in leukocytes and platelets MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-29 US disclosed
EP-0476645-A1 Calcium uptake inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1992-03-25 EP disclosed
US-4818096-A SUNGLASSES; BENZO OR NAPHTHOPYRANS WITH NITROGEN CONTAINING SUBSTITUENTS THE PLESSEY COMPANY PLC (GB) 1989-04-04 US disclosed
EP-0250193-A2 Photoreactive lenses GEC-MARCONI LIMITED (GB) 1987-12-23 EP disclosed