SCHEMBL9136294

SCHEMBL9136294

O=C1CCCN(C(c2ccccc2)(c2ccccc2)c2ccccc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2B6 P20813 1/20 0.42
ALOX5 P09917 2/20 0.35
POLB P06746 1/20 0.33
KMT2A Q03164 3/20 0.32
MEN1 O00255 2/20 0.32
CYP2C9 P11712 2/20 0.32
ALDH1A1 P00352 2/20 0.32
HSD17B10 Q99714 2/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
KDM4E B2RXH2 1/20 0.32
USP2 O75604 1/20 0.32
CYP1A2 P05177 1/20 0.32
BCHE P06276 1/20 0.32
CFTR P13569 1/20 0.32
ALOX15 P16050 1/20 0.32
ACHE P22303 1/20 0.32
HKDC1 Q2TB90 1/20 0.32
GOPC Q9HD26 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CHRM3 P20309 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3744280 0.93 CYP2B6 (0.38) CYP2B6ALOX5POLBKMT2AMEN1
SCHEMBL4400626 0.86 CYP2B6 (0.42) CYP2B6ALOX5KMT2AMEN1CYP2C9
SCHEMBL1528523 0.81 CYP2B6 (0.36) CYP2B6ALOX5POLBKMT2AMEN1
SCHEMBL27753492 0.80 CYP2B6 (0.54) CYP2B6KMT2AMEN1CYP2C9ALDH1A1
SCHEMBL2392136 0.80 CYP2B6 (0.59) CYP2B6KMT2AMEN1CYP2C9ALDH1A1
Chlorotriphenylmethane SCHEMBL8598442 0.79 CYP2B6 (0.37) CYP2B6ALOX5CYP1A2
SCHEMBL2491599 0.78 CYP2B6 (0.63) CYP2B6KMT2AMEN1CYP2C9KDM4E
SCHEMBL19296941 0.78 CYP2B6 (0.63) CYP2B6KMT2AMEN1CYP2C9KDM4E
SCHEMBL9650536 0.76 CYP2B6 (0.46) CYP2B6ALDH1A1KDM4ECHRM3LMNA
SCHEMBL3707837 0.74 CYP2B6 (0.63) CYP2B6POLBKMT2AMEN1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5466687-A Anticholesterol agents DR. KARL THOMAE GMBH (DE) 1995-11-14 US disclosed
EP-0596326-B1 Arylidene-1-azacycloalkanes and arylalkyl-1-azacycloalkanes, their salts, medicaments containing the same, use thereof and precesses for their production THOMAE GMBH DR K (DE) 1995-08-23 EP disclosed
EP-0596326-A1 Arylidene-1-azacycloalkanes and arylalkyl-1-azacycloalkanes, their salts, medicaments containing the same, use thereof and precesses for their production Dr. Karl Thomae GmbH (DE) 1994-05-11 EP disclosed