SCHEMBL9136295

SCHEMBL9136295

CCOC(=O)c1ccc(-c2c(C)[nH]c(C)cc2=O)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.58
ALDH1A1 P00352 4/20 0.58
HPGD P15428 4/20 0.58
POLB P06746 1/20 0.58
MAPK1 P28482 1/20 0.58
HSD17B10 Q99714 1/20 0.58
CA12 O43570 2/20 0.48
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CA7 P43166 2/20 0.48
CA9 Q16790 2/20 0.48
CA14 Q9ULX7 2/20 0.48
ESR1 P03372 1/20 0.47
ESR2 Q92731 1/20 0.47
SLC11A2 P49281 1/20 0.47
HCRTR1 O43613 1/20 0.47
CYP1A2 P05177 2/20 0.46
LMNA P02545 1/20 0.46
CYP3A4 P08684 1/20 0.46
MAOA P21397 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9135228 0.85 POLB (0.54) KDM4EALDH1A1HPGDPOLBMAPK1
SCHEMBL8597367 0.81 CA12 (0.51) KDM4EALDH1A1HPGDPOLBMAPK1
SCHEMBL11233586 0.78 CA1 (0.68) KDM4EALDH1A1HPGDCA12CA1
SCHEMBL9139438 0.77 TNKS (0.46) KDM4EALDH1A1HPGDPOLBMAPK1
SCHEMBL9455121 0.75 ALDH1A1 (0.46) KDM4EALDH1A1HPGDPOLBMAPK1
SCHEMBL16351874 0.75 CA1 (0.73) KDM4EALDH1A1HPGDCA12CA1
SCHEMBL1965326 0.75 CA1 (0.73) KDM4EALDH1A1HPGDCA12CA1
SCHEMBL3189642 0.74 ALDH1A1 (0.61) KDM4EALDH1A1HPGDPOLBMAPK1
SCHEMBL25911102 0.73 KDM4E (0.80) KDM4EALDH1A1HPGDPOLBMAPK1
SCHEMBL87450 0.73 CA1 (0.83) ALDH1A1HPGDCA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5380730-A Angiotensin antagonist IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1995-01-10 US disclosed
US-5236936-A Treating hypertension, congestive heart failure IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-08-17 US disclosed
EP-0499416-A2 Pyridine compounds as angiotensin II antagonists, processes for their preparation and pharmaceutical compositions containing them ZENECA LIMITED (GB) 1992-08-19 EP disclosed