SCHEMBL9136357

SCHEMBL9136357

C[C@@H](NC(=O)OCc1ccccc1)C(=O)NCCNC(=O)[C@@H](C)NC(=O)OCc1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSK P43235 10/20 0.62
CYP1A2 P05177 1/20 0.62
TPSAB1 Q15661 2/20 0.61
PLG P00747 1/20 0.61
PRSS1 P07477 1/20 0.61
CTSS P25774 6/20 0.57
CTSL P07711 4/20 0.57
CTSB P07858 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11702018 0.93 CYP1A2 (0.58) CTSKCYP1A2TPSAB1PLGPRSS1
SCHEMBL8502694 0.93 CYP1A2 (0.58) CTSKCYP1A2TPSAB1PLGPRSS1
SCHEMBL10954836 0.93 CA5A (0.62) CTSKCYP1A2TPSAB1PLGPRSS1
SCHEMBL10957418 0.93 CYP1A2 (0.58) CTSKCYP1A2TPSAB1PLGPRSS1
SCHEMBL15318479 0.93 CA5A (0.62) CTSKCYP1A2TPSAB1PLGPRSS1
SCHEMBL4075738 0.91 CYP1A2 (0.62) CTSKCYP1A2TPSAB1PLGPRSS1
SCHEMBL10954266 0.91 CA5A (0.60) CTSKCYP1A2TPSAB1PLGPRSS1
SCHEMBL12294550 0.91 CYP2D6 (0.62) CTSKCYP1A2TPSAB1PLGPRSS1
SCHEMBL30387033 0.90 SYK (0.63) CTSKCYP1A2TPSAB1PLGPRSS1
SCHEMBL10953796 0.90 CYP1A2 (0.61) CTSKCYP1A2TPSAB1PLGPRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5461176-A Reacting alanine methyl ester with oxalyl chloride, treating with ammonia in methanol, reducing amides with diborane in tetrahydrofuran, neutralizing with sodium ethoxide to yield free amine THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-10-24 US disclosed