SCHEMBL9140293

SCHEMBL9140293

CCOC(=O)c1ccc(/C=C(\C)c2ccc3c(c2)CCC(C)CS3)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARG P13631 9/20 0.45
RARB P10826 8/20 0.45
RARA P10276 6/20 0.45
MAPT P10636 3/20 0.38
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 2/20 0.37
NPC1 O15118 2/20 0.37
ALDH1A1 P00352 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
DRD3 P35462 2/20 0.37
DRD2 P14416 1/20 0.37
LMNA P02545 2/20 0.36
KDM4E B2RXH2 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
ESR1 P03372 1/20 0.36
CA7 P43166 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9140302 1.00 RARG (0.45) RARGRARBRARAMAPTHPGD
SCHEMBL26471776 0.87 RARG (0.43) RARGRARBRARAMAPTHPGD
SCHEMBL9145537 0.86 RARG (0.48) RARGRARBRARAHPGDHTT
SCHEMBL9145541 0.86 RARG (0.48) RARGRARBRARAHPGDHTT
SCHEMBL8460903 0.86 DRD3 (0.44) RARGRARBRARAMAPTHPGD
SCHEMBL8460900 0.86 DRD3 (0.44) RARGRARBRARAMAPTHPGD
SCHEMBL8457141 0.85 RARG (0.54) RARGRARBRARARAB9ANPC1
SCHEMBL8457147 0.85 RARG (0.54) RARGRARBRARARAB9ANPC1
SCHEMBL9144382 0.83 RARB (0.51) RARGRARBRARAMAPTHPGD
SCHEMBL9144389 0.83 RARB (0.51) RARGRARBRARAMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5420273-A Skin disorders and antitumor agents HOFFMAN-LA ROCHE INC. (US) 1995-05-30 US disclosed
US-5164387-A Antitumor agents, skin disorders, antiinflammatory agents HOFFMANN-LAROCHE INC. (US) 1992-11-17 US disclosed
US-5037825-A Useful In The Treatment Of Neoplasms, Dermatoses And Aging Of The Skin HOFFMANN-LA ROCHE INC. (US) 1991-08-06 US disclosed