SCHEMBL8460903

SCHEMBL8460903

CCOC(=O)c1ccc(C=C(C)c2ccc3c(c2)CCC(C)CC3)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 2/20 0.44
DRD2 P14416 1/20 0.44
RARG P13631 8/20 0.41
RARB P10826 7/20 0.41
RARA P10276 5/20 0.41
HPGD P15428 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 3/20 0.40
MAPT P10636 2/20 0.40
NPC1 O15118 2/20 0.40
ALDH1A1 P00352 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
ESR1 P03372 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
ESR2 Q92731 1/20 0.40
CA14 Q9ULX7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8460900 1.00 DRD3 (0.44) DRD3DRD2RARGRARBRARA
SCHEMBL9419049 0.87 HPGD (0.44) DRD3DRD2RARGRARBRARA
SCHEMBL9419050 0.87 HPGD (0.44) DRD3DRD2RARGRARBRARA
SCHEMBL9140302 0.86 RARG (0.45) DRD3DRD2RARGRARBRARA
SCHEMBL9140293 0.86 RARG (0.45) DRD3DRD2RARGRARBRARA
SCHEMBL8458507 0.86 HTT (0.43) RARGRARBRARAHPGDHTT
SCHEMBL8458513 0.86 HTT (0.43) RARGRARBRARAHPGDHTT
SCHEMBL7223039 0.84 RARB (0.48) RARGRARBRARAHPGDHTT
SCHEMBL9419019 0.84 RARB (0.48) RARGRARBRARAHPGDHTT
SCHEMBL9418999 0.84 RARB (0.46) RARGRARBRARAHPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0315071-B1 Benzocyclohepten derivatives, their preparation and utilisation for pharmaceutics HOFFMANN LA ROCHE (CH) 1994-07-20 EP claimed
WO-1999048529-A1 RETINOID-GLITAZONE COMBINATIONS WARNER-LAMBERT COMPANY (US) 1999-09-30 WO disclosed
EP-0808159-A1 USE OR RETINOIDS TO LOWER PLASMA LEVELS OF LIPOPROTEIN (a) WARNER-LAMBERT COMPANY (US) 1997-11-26 EP disclosed
WO-1996024344-A1 USE OF RETINOIDS TO LOWER PLASMA LEVELS OF LIPOPROTEIN (a) WARNER-LAMBERT COMPANY (US) 1996-08-15 WO disclosed
US-5489611-A ADMINISTERING A RETINOID COMPOUND WARNER-LAMBERT COMPANY (US) 1996-02-06 US disclosed