SCHEMBL9140451

SCHEMBL9140451

CCCCc1cc(N)n[nH]1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 6/20 0.54
HCAR3 P49019 4/20 0.54
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
MAPT P10636 1/20 0.49
GFER P55789 1/20 0.49
TP53 P04637 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
TSHR P16473 1/20 0.42
NOS2 P35228 1/20 0.42
HRH3 Q9Y5N1 1/20 0.41
MITF O75030 1/20 0.40
ALDH1A1 P00352 1/20 0.40
KMT2A Q03164 1/20 0.40
GAA P10253 1/20 0.39
HSD17B10 Q99714 1/20 0.39
DAO P14920 1/20 0.39
GPR84 Q9NQS5 2/20 0.39
DYRK1A Q13627 1/20 0.36
GABRP O00591 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2865249 0.94 HCAR2 (0.56) HCAR2HCAR3NPC1RAB9AMAPT
SCHEMBL8512535 0.92 HCAR2 (0.57) HCAR2HCAR3NPC1RAB9AMAPT
SCHEMBL1706467 0.88
Hydrochloric Acid SCHEMBL1707357 0.86 NPC1 (0.54) HCAR2HCAR3NPC1RAB9AMAPT
SCHEMBL4011081 0.82 GAA (0.42) HCAR2HCAR3NPC1RAB9AMAPT
SCHEMBL4161900 0.79 HCAR2 (0.45) HCAR2HCAR3NPC1RAB9AMAPT
SCHEMBL174227 0.79
SCHEMBL27396391 0.78 DAO (0.41) HCAR2HCAR3NPC1RAB9AMAPT
SCHEMBL23891666 0.78 HCAR2 (0.56) HCAR2HCAR3NPC1RAB9ANOS2
SCHEMBL2765959 0.78 HCAR2 (0.56) HCAR2HCAR3NOS2HRH3DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5475114-A Angiotensin-11 antagonist; therapeutical agent used for treating hypertension and chronic heart failure YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1995-12-12 US disclosed
EP-0646584-A1 PYRAZOLOTRIAZOLE DERIVATIVE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-04-05 EP disclosed
CN-1069978-A Pyrazolotriazole derivatives YAMANOUCHI PHARMA CO LTD (JP) 1993-03-17 CN disclosed