SCHEMBL9145751

SCHEMBL9145751

COC(=O)c1ccc(C=C(C)c2ccc3c(c2)OC(C)(C)O3)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 12/20 0.64
RARG P13631 12/20 0.64
RARA P10276 11/20 0.61
ALDH1A1 P00352 2/20 0.44
RAB9A P51151 4/20 0.41
NPC1 O15118 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
RXRA P19793 2/20 0.41
POLB P06746 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CYP26A1 O43174 1/20 0.41
GMNN O75496 1/20 0.41
USP2 O75604 1/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
NFKB1 P19838 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9145742 1.00 RARB (0.64) RARBRARGRARAALDH1A1RAB9A
SCHEMBL8522590 0.85 RARG (0.62) RARBRARGRARAALDH1A1RAB9A
SCHEMBL8522592 0.85 RARG (0.62) RARBRARGRARAALDH1A1RAB9A
SCHEMBL24401018 0.83 ALOX5 (0.50) RARBRARGALDH1A1RAB9ANPC1
SCHEMBL26722153 0.78 RARB (1.00) RARBRARGRARAALDH1A1RAB9A
SCHEMBL10556851 0.76 RARB (1.00) RARBRARGRARAALDH1A1RAB9A
SCHEMBL10556841 0.76 RARB (1.00) RARBRARGRARAALDH1A1RAB9A
SCHEMBL12367125 0.75 MAPT (0.41) RARBRARGRARAALDH1A1RAB9A
SCHEMBL9142620 0.74 RARB (0.61) RARBRARGRARAALDH1A1RAB9A
SCHEMBL9142618 0.74 RARB (0.61) RARBRARGRARAALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0350846-B1 Condensed heterocyclic compounds and their use in therapy HOFFMANN LA ROCHE (CH) 1995-10-11 EP claimed
US-5420273-A Skin disorders and antitumor agents HOFFMAN-LA ROCHE INC. (US) 1995-05-30 US disclosed
US-5300522-A Treating inflammatory, allergic, rheumatic, immunological disorders HOFFMANN-LA ROCHE INC. (US) 1994-04-05 US disclosed
US-5164387-A Antitumor agents, skin disorders, antiinflammatory agents HOFFMANN-LAROCHE INC. (US) 1992-11-17 US disclosed
US-5037825-A Useful In The Treatment Of Neoplasms, Dermatoses And Aging Of The Skin HOFFMANN-LA ROCHE INC. (US) 1991-08-06 US disclosed