SCHEMBL9147176

SCHEMBL9147176

N#Cc1cc(-c2cnc(N)nc2N)ccc1Cl

nearest known ligand 0.68

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DHFR P00374 6/20 0.68
ADORA1 P30542 5/20 0.47
ADORA2A P29274 5/20 0.42
FGFR1 P11362 1/20 0.42
SRC P12931 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
CSNK1A1 P48729 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
MAPK14 Q16539 1/20 0.40
PTPN11 Q06124 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1388267 0.82 DHFR (1.00) DHFRADORA1ADORA2AFGFR1SRC
SCHEMBL1388741 0.80 DHFR (0.79) DHFRADORA1ADORA2AFGFR1SRC
SCHEMBL1388760 0.75 DHFR (0.74) DHFRADORA1ADORA2AFGFR1SRC
SCHEMBL1388517 0.75 DHFR (0.74) DHFRADORA1ADORA2AFGFR1SRC
SCHEMBL1388506 0.73 DHFR (0.67) DHFRLMNA
SCHEMBL29913206 0.73 DHFR (0.67) DHFRLMNA
SCHEMBL1388763 0.72 DHFR (1.00) DHFRADORA1ALDH1A1
SCHEMBL7273497 0.72 DHFR (0.70) DHFRADORA1ADORA2AFGFR1SRC
SCHEMBL1388629 0.71 ADORA1 (0.70) DHFRADORA1ADORA2A
SCHEMBL1388616 0.71 DHFR (0.63) DHFRADORA1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0674627-A1 PYRIMIDINE, PYRIDINE, PTERIDINONE AND INDAZOLE DERIVATIVES AS ENZYME INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1995-10-04 EP disclosed
WO-1994014780-A1 PYRIMIDINE, PYRIDINE, PTERIDINONE AND INDAZOLE DERIVATIVES AS ENZYME INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1994-07-07 WO disclosed