SCHEMBL9149374

SCHEMBL9149374

O=C(O)CC1OCCc2cc3c(cc21)OCO3

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
GLA P06280 2/20 0.40
HPGD P15428 2/20 0.40
CASP1 P29466 2/20 0.40
CASP7 P55210 2/20 0.40
HSD17B10 Q99714 2/20 0.40
CYP2D6 P10635 1/20 0.40
GAA P10253 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.37
ADRA1A P35348 3/20 0.37
DRD2 P14416 1/20 0.37
DRD1 P21728 1/20 0.37
ADRA2A P08913 3/20 0.36
ADRA2B P18089 3/20 0.36
ADRA2C P18825 3/20 0.36
ADRA1D P25100 2/20 0.36
ADRA1B P35368 2/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11224140 0.79 KDM4E (0.41) KDM4EALDH1A1GLAHPGDCASP1
SCHEMBL11225616 0.77 KDM4E (0.39) KDM4EALDH1A1GLAHPGDCASP1
SCHEMBL8550598 0.75 GAA (0.43) KDM4EALDH1A1HSD17B10GAAL3MBTL1
SCHEMBL19813046 0.75 TAAR1 (0.55) KDM4EALDH1A1GLAHPGDCASP1
SCHEMBL30360731 0.75 TAAR1 (0.55) KDM4EALDH1A1GLAHPGDCASP1
SCHEMBL19812985 0.75 TAAR1 (0.55) KDM4EALDH1A1GLAHPGDCASP1
SCHEMBL32670646 0.75 TAAR1 (0.55) KDM4EALDH1A1GLAHPGDCASP1
SCHEMBL19812870 0.75 TAAR1 (0.55) KDM4EALDH1A1GLAHPGDCASP1
SCHEMBL5093605 0.74 MAPT (0.43) ALDH1A1GAAL3MBTL1APEX1
SCHEMBL5090662 0.74 MAPT (0.43) ALDH1A1GAAL3MBTL1APEX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5475024-A Useful in treating liver disease EISAI CO., LTD. (JP) 1995-12-12 US disclosed
US-5292901-A Benzodioxole derivatives EISAI CO., LTD. (JP) 1994-03-08 US disclosed
EP-0281098-B1 BENZODIOXOLE DERIVATIVES, COMPOSITIONS COMPRISING THE SAME, AND THE USE OF THE SAME FOR THE MANUFACTURE OF MEDICAMENTS Eisai Co., Ltd. (JP) 1992-11-25 EP disclosed
US-5110956-A Liver disorders EISAI CO., LTD. (JP) 1992-05-05 US disclosed
EP-0281098-A1 Benzodioxole derivatives, compositions comprising the same, and the use of the same for the manufacture of medicaments Eisai Co., Ltd. (JP) 1988-09-07 EP disclosed