SCHEMBL11225616

SCHEMBL11225616

ClCCC1OCCc2cc3c(cc21)OCO3

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
GLA P06280 2/20 0.39
HPGD P15428 2/20 0.39
CASP1 P29466 2/20 0.39
CASP7 P55210 2/20 0.39
HSD17B10 Q99714 2/20 0.39
CYP2D6 P10635 1/20 0.39
ADRA1A P35348 1/20 0.38
GAA P10253 1/20 0.38
DRD2 P14416 1/20 0.38
DRD1 P21728 1/20 0.38
CYP3A4 P08684 1/20 0.36
HTR1A P08908 1/20 0.36
CHRNA7 P36544 3/20 0.36
ADRA2A P08913 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11220977 0.91 KDM4E (0.38) KDM4EALDH1A1GLAHPGDCASP1
SCHEMBL11224140 0.81 KDM4E (0.41) KDM4EALDH1A1GLAHPGDCASP1
SCHEMBL19813046 0.78 TAAR1 (0.55) KDM4EALDH1A1GLAHPGDCASP1
SCHEMBL30360731 0.78 TAAR1 (0.55) KDM4EALDH1A1GLAHPGDCASP1
SCHEMBL19812870 0.78 TAAR1 (0.55) KDM4EALDH1A1GLAHPGDCASP1
SCHEMBL19812985 0.78 TAAR1 (0.55) KDM4EALDH1A1GLAHPGDCASP1
SCHEMBL32670646 0.78 TAAR1 (0.55) KDM4EALDH1A1GLAHPGDCASP1
SCHEMBL9149374 0.77 KDM4E (0.40) KDM4EALDH1A1GLAHPGDCASP1
SCHEMBL9688216 0.75 KCNN2 (0.43) KDM4EALDH1A1HSD17B10CYP2D6
SCHEMBL11226052 0.74 KDM4E (0.34) KDM4EALDH1A1GLAHPGDCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4352805-A BENZOXEPINE DERIVATIVES THE UPJOHN COMPANY (US) 1982-10-05 US disclosed
US-4312868-A HYPOTENSIVE, ANTIPSYCHOTIC THE UPJOHN COMPANY (US) 1982-01-26 US disclosed
US-4251526-A HYPOTENSIVE AGENTS AND ANTIPSYCHOTIC PHARMACIA & UPJOHN COMPANY 1981-02-17 US disclosed
US-4250175-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS PHARMACIA & UPJOHN COMPANY 1981-02-10 US disclosed
US-4250181-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-02-10 US disclosed
US-4247553-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-01-27 US disclosed
US-4179510-A ISOCHROMANS AND 2-BENZOXEPINS THE UPJOHN COMPANY (US) 1979-12-18 US disclosed
US-4166062-A HYPOTENSIVE AGENTS, CNS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1979-08-28 US disclosed
US-4153612-A 2-Benzoxepins THE UPJOHN COMPANY (US) 1979-05-08 US disclosed