SCHEMBL9150745

SCHEMBL9150745

Cc1nsc(C2CN3CCCC2C3)n1

nearest known ligand 0.54

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9147996 0.91 CHRM2 (0.51) CHRM2
Oxalic Acid SCHEMBL9151057 0.86 CHRM2 (0.45) CHRM2
SCHEMBL9151214 0.83 CHRM1 (0.43) CHRM2
SCHEMBL9150768 0.83 CHRNA7 (0.42) CHRM2
Oxalic Acid SCHEMBL9148594 0.78 CHRNA7 (0.40) CHRM2
SCHEMBL9149572 0.75 CHRM2 (0.35) CHRM2
SCHEMBL9151072 0.74 DPP4 (0.35) CHRM2
SCHEMBL9148633 0.73 CHRM2 (0.53) CHRM2
SCHEMBL9147958 0.72 CHRM2 (0.41) CHRM2
SCHEMBL9152399 0.72 CHRM2 (0.41) CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0307142-B1 Thiadiazoles useful in the treatment of senile dementia MERCK SHARP & DOHME (GB) 1994-09-14 EP claimed
US-5405853-A Potent muscarinic agonists having good central nervous system penetrability MERCK SHARPE & DOHME LTD. (GB) 1995-04-11 US disclosed
EP-0307142-B1 Thiadiazoles useful in the treatment of senile dementia MERCK SHARP & DOHME (GB) 1994-09-14 EP disclosed
EP-0307142-A1 Thiadiazoles useful in the treatment of senile dementia MERCK SHARP & DOHME LTD. (GB) 1989-03-15 EP disclosed