SCHEMBL9152227

SCHEMBL9152227

Nc1nsc(C2CN3CCC2C(O)C3)n1

nearest known ligand 0.35

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9151670 0.86
SCHEMBL9151072 0.84 DPP4 (0.35) CHRM2
SCHEMBL9151515 0.82 CHRM2 (0.35) CHRM2CHRM1
SCHEMBL9148633 0.78 CHRM2 (0.53) CHRM2CHRM1
SCHEMBL9152478 0.76 CHRNA7 (0.43) CHRM2CHRM1
SCHEMBL9151214 0.73 CHRM1 (0.43) CHRM2CHRM1
SCHEMBL9369971 0.72 CHRM2 (0.65) CHRM2CHRM1
SCHEMBL9150021 0.71
SCHEMBL9149591 0.70 DPP4 (0.32)
SCHEMBL9149572 0.68 CHRM2 (0.35) CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5405853-A Potent muscarinic agonists having good central nervous system penetrability MERCK SHARPE & DOHME LTD. (GB) 1995-04-11 US claimed
EP-0307142-B1 Thiadiazoles useful in the treatment of senile dementia MERCK SHARP & DOHME (GB) 1994-09-14 EP claimed
EP-0307142-A1 Thiadiazoles useful in the treatment of senile dementia MERCK SHARP & DOHME LTD. (GB) 1989-03-15 EP claimed
US-5405853-A Potent muscarinic agonists having good central nervous system penetrability MERCK SHARPE & DOHME LTD. (GB) 1995-04-11 US disclosed
EP-0307142-B1 Thiadiazoles useful in the treatment of senile dementia MERCK SHARP & DOHME (GB) 1994-09-14 EP disclosed
EP-0307142-A1 Thiadiazoles useful in the treatment of senile dementia MERCK SHARP & DOHME LTD. (GB) 1989-03-15 EP disclosed