SCHEMBL9155754

SCHEMBL9155754

COc1ccc(-c2ccc(-c3ccc(C(F)(F)F)nc3)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.49
NT5E P21589 1/20 0.49
PDE10A Q9Y233 1/20 0.48
PTGS1 P23219 2/20 0.48
PTGS2 P35354 2/20 0.48
CYP11B1 P15538 1/20 0.47
CYP11B2 P19099 1/20 0.47
TRPV4 Q9HBA0 1/20 0.46
SYK P43405 1/20 0.45
TP53 P04637 2/20 0.44
KMT2A Q03164 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
USP2 O75604 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
SCN5A Q14524 1/20 0.44
PDGFRB P09619 1/20 0.44
PDGFRA P16234 1/20 0.44
MAP4K4 O95819 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31414063 1.00 KDM4E (0.49) KDM4ENT5EPDE10APTGS1PTGS2
SCHEMBL929327 0.85 TRPV4 (0.52) KDM4ENT5EPDE10APTGS1PTGS2
SCHEMBL31130640 0.83 TRPV4 (0.50) KDM4ENT5EPDE10APTGS1PTGS2
SCHEMBL9253133 0.83 GRM5 (0.47) KDM4EPTGS1PTGS2TRPV4TP53
SCHEMBL9159912 0.83 GRM5 (0.47) KDM4EPTGS1PTGS2TRPV4TP53
SCHEMBL9160877 0.80 CYP2D6 (0.48) KDM4ETP53SMN1; SMN2ALDH1A1HPGD
SCHEMBL9160694 0.80 CYP2D6 (0.48) KDM4ETP53SMN1; SMN2ALDH1A1HPGD
SCHEMBL9154037 0.80 CYP2D6 (0.55) KDM4EPTGS1PTGS2SMN1; SMN2GRM5
SCHEMBL9158809 0.80 CYP2D6 (0.55) KDM4EPTGS1PTGS2SMN1; SMN2GRM5
SCHEMBL9766710 0.80 CYP2D6 (0.42) KDM4EKMT2AALDH1A1HPGDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445248-B1 PYRIDINE DERIVATIVES MERCK PATENT GMBH (DE) 1995-03-08 EP disclosed
US-5205962-A Stable liquid crystals MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1993-04-27 US disclosed