SCHEMBL9156922

SCHEMBL9156922

O=C1CC=C(Cl)c2c1[nH]c(=O)c1cccn21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 12/20 0.43
TP53 P04637 1/20 0.38
CDC7 O00311 2/20 0.32
PLK4 O00444 2/20 0.32
MAPK13 O15264 2/20 0.32
PDPK1 O15530 2/20 0.32
DYRK3 O43781 2/20 0.32
ERBB2 P04626 2/20 0.32
PRKCG P05129 2/20 0.32
ROS1 P08922 2/20 0.32
KIT P10721 2/20 0.32
SRC P12931 2/20 0.32
PHKG2 P15735 2/20 0.32
AKT1 P31749 2/20 0.32
AKT2 P31751 2/20 0.32
MATK P42679 2/20 0.32
MAPKAPK2 P49137 2/20 0.32
BLK P51451 2/20 0.32
IRAK1 P51617 2/20 0.32
NEK4 P51957 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9155013 0.71 PARP1 (0.45) PARP1TP53CDC7PLK4MAPK13
SCHEMBL9155368 0.63 PARP1 (0.43) PARP1TP53CDC7PLK4MAPK13
SCHEMBL1133601 0.61 PARP1 (1.00) PARP1TP53CDC7PLK4MAPK13
SCHEMBL29673205 0.61 PARP1 (1.00) PARP1TP53CDC7PLK4MAPK13
SCHEMBL8569594 0.61 TP53 (0.68) PARP1TP53CDC7PLK4MAPK13
SCHEMBL2429766 0.61 PARP1 (0.65) PARP1TP53CDC7PLK4MAPK13
SCHEMBL9415441 0.61 PARP1 (0.60) PARP1TP53CDC7PLK4MAPK13
SCHEMBL21405585 0.60 PARP1 (0.50) PARP1TP53CDC7PLK4MAPK13
SCHEMBL30929174 0.60 PARP1 (0.55) PARP1TP53CDC7PLK4MAPK13
SCHEMBL8565857 0.59 PARP1 (0.53) PARP1TP53CDC7PLK4MAPK13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5405847-A Antiallergic, antiasthmatic, anxiolytic, hypotensive agents ASTA MEDICA AKTIENGESELLSCHAFT (DE) 1995-04-11 US disclosed