SCHEMBL9415441

SCHEMBL9415441

O=c1[nH]c2cccc(Cl)c2n2cccc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 11/20 0.60
TP53 P04637 1/20 0.48
PSMB8 P28062 1/20 0.45
DAO P14920 1/20 0.41
MAP4K4 O95819 2/20 0.40
TAOK1 Q7L7X3 2/20 0.40
PBK Q96KB5 1/20 0.40
SLK Q9H2G2 1/20 0.40
GRIN2D O15399 2/20 0.40
GRIN3B O60391 2/20 0.40
GRIN1 Q05586 2/20 0.40
GRIN2A Q12879 2/20 0.40
GRIN2B Q13224 2/20 0.40
GRIN2C Q14957 2/20 0.40
GRIN3A Q8TCU5 2/20 0.40
ALDH1A1 P00352 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
PLA2G10 O15496 1/20 0.39
MGAM O43451 1/20 0.39
PLA2G2A P14555 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14361434 0.81 PARP1 (0.60) PARP1TP53DAOMAP4K4TAOK1
SCHEMBL29673205 0.75 PARP1 (1.00) PARP1TP53DAOMAP4K4TAOK1
SCHEMBL1133601 0.75 PARP1 (1.00) PARP1TP53DAOMAP4K4TAOK1
SCHEMBL30273115 0.72 PSMB8 (0.40) PARP1PSMB8DAOMAP4K4TAOK1
SCHEMBL8569594 0.71 TP53 (0.68) PARP1TP53MAP4K4TAOK1PBK
SCHEMBL2429766 0.71 PARP1 (0.65) PARP1TP53DAOMAP4K4TAOK1
SCHEMBL10503087 0.70 PSMB8 (0.60) PSMB8DAOGRIN2DGRIN3BGRIN1
SCHEMBL7276765 0.70 PARP1 (0.69) PARP1TP53DAOGRIN2DGRIN3B
SCHEMBL8565857 0.69 PARP1 (0.53) PARP1TP53MAP4K4TAOK1PBK
SCHEMBL30809703 0.68 PDE2A (0.67) PARP1TP53DAOGRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0584487-A2 4,5-Dihydro-4-oxopyrrolo (1,2-a) quinoxalines and aza-analoges and process for their preparation ASTA Medica Aktiengesellschaft (DE) 1994-03-02 EP disclosed