SCHEMBL9157229

SCHEMBL9157229

CCCCCOc1ccc(-c2ccc(C#Cc3ccc(F)nc3F)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 6/20 0.44
CYP3A4 P08684 4/20 0.44
HPGD P15428 4/20 0.43
KDM4E B2RXH2 4/20 0.43
ALDH1A1 P00352 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
HTT P42858 1/20 0.43
RARB P10826 3/20 0.42
MCHR1 Q99705 2/20 0.40
CYP19A1 P11511 5/20 0.40
CYP2C9 P11712 5/20 0.40
CYP2C19 P33261 5/20 0.40
CYP1A2 P05177 4/20 0.40
NR5A1 Q13285 1/20 0.39
RAB9A P51151 4/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
LTA4H P09960 1/20 0.38
NPC1 O15118 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9157311 0.97 CYP2D6 (0.47) CYP2D6CYP3A4HPGDKDM4EALDH1A1
SCHEMBL9158961 0.96 NR5A1 (0.42) CYP2D6CYP3A4HPGDKDM4EALDH1A1
SCHEMBL9158222 0.94 ACACB (0.40) CYP2D6CYP3A4HPGDKDM4EALDH1A1
SCHEMBL9157720 0.92 MCHR1 (0.42) CYP2D6CYP3A4HPGDKDM4EALDH1A1
SCHEMBL9766659 0.92 CYP2D6 (0.42) CYP2D6CYP3A4HPGDKDM4EALDH1A1
SCHEMBL9154867 0.88 ACACB (0.41) HTTLMNAHSD17B10
SCHEMBL9158464 0.87 NQO1 (0.39) HPGDKDM4EALDH1A1MCHR1RAB9A
SCHEMBL9766674 0.86 MCHR1 (0.39) HPGDKDM4EALDH1A1L3MBTL1HTT
SCHEMBL9156038 0.84 HSD17B10 (0.49) CYP3A4HPGDKDM4EALDH1A1RARB
SCHEMBL9159722 0.83 NQO1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445248-B1 PYRIDINE DERIVATIVES MERCK PATENT GMBH (DE) 1995-03-08 EP disclosed
US-5205962-A Stable liquid crystals MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1993-04-27 US disclosed
EP-0445248-A1 PYRIDINE DERIVATIVES. MERCK PATENT GMBH (DE) 1991-09-11 EP disclosed
WO-1991004248-A1 PYRIDINE DERIVATIVES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1991-04-04 WO disclosed