SCHEMBL9766659

SCHEMBL9766659

CCCCOc1ccc(-c2ccc(C#Cc3ccc(F)nc3F)cc2)cc1.CCCOc1ccc(-c2ccc(C#Cc3ccc(F)nc3F)cc2)cc1.CCOc1ccc(-c2ccc(C#Cc3ccc(F)nc3F)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 6/20 0.42
CYP3A4 P08684 4/20 0.42
MCHR1 Q99705 2/20 0.38
CYP19A1 P11511 5/20 0.38
CYP2C9 P11712 5/20 0.38
CYP2C19 P33261 5/20 0.38
CYP1A2 P05177 5/20 0.38
ACACB O00763 1/20 0.38
ACACA Q13085 1/20 0.38
GAA P10253 2/20 0.37
RAB9A P51151 6/20 0.36
HPGD P15428 5/20 0.36
ALDH1A1 P00352 4/20 0.36
SMN1; SMN2 Q16637 4/20 0.36
ALOX12 P18054 1/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
KDM4E B2RXH2 4/20 0.36
TP53 P04637 2/20 0.36
MAPT P10636 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9157720 0.94 MCHR1 (0.42) CYP2D6CYP3A4MCHR1CYP1A2ACACB
SCHEMBL9157311 0.94 CYP2D6 (0.47) CYP2D6CYP3A4MCHR1CYP19A1CYP2C9
SCHEMBL9157229 0.92 CYP2D6 (0.44) CYP2D6CYP3A4MCHR1CYP19A1CYP2C9
SCHEMBL9158464 0.92 NQO1 (0.39) MCHR1ACACBGAARAB9AHPGD
SCHEMBL9158222 0.90 ACACB (0.40) CYP2D6CYP3A4CYP19A1CYP2C9CYP2C19
SCHEMBL9154867 0.90 ACACB (0.41) ACACBLMNAHTTHSD17B10
SCHEMBL9766674 0.90 MCHR1 (0.39) MCHR1ACACBHPGDALDH1A1KDM4E
SCHEMBL9158961 0.88 NR5A1 (0.42) CYP2D6CYP3A4CYP19A1CYP2C9CYP2C19
SCHEMBL9159722 0.88 NQO1 (0.42) ACACB
SCHEMBL9155712 0.79 TSHR (0.43) RAB9AALDH1A1SMN1; SMN2TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445248-A1 PYRIDINE DERIVATIVES. MERCK PATENT GMBH (DE) 1991-09-11 EP disclosed