SCHEMBL9157458

SCHEMBL9157458

COC(=O)c1cccc(NC(=O)c2cn(C)c3ccccc23)c1

nearest known ligand 0.76

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 3/20 0.76
NR4A2 P43354 1/20 0.61
SRC P12931 1/20 0.61
RAB9A P51151 3/20 0.60
MAOB P27338 3/20 0.58
EP300 Q09472 1/20 0.58
TSHR P16473 3/20 0.56
ALDH1A1 P00352 2/20 0.56
NPSR1 Q6W5P4 2/20 0.56
SMN1; SMN2 Q16637 3/20 0.53
TP53 P04637 2/20 0.53
MAPT P10636 2/20 0.53
HIF1A Q16665 1/20 0.53
LMNA P02545 1/20 0.52
POLB P06746 2/20 0.51
NPC1 O15118 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9158175 0.86 NR4A2 (0.66) CREBBPNR4A2SRCRAB9AMAOB
SCHEMBL28624532 0.86 CREBBP (1.00) CREBBPSRCRAB9AEP300
SCHEMBL6005094 0.82 MAOB (0.61) CREBBPNR4A2MAOBEP300ALDH1A1
SCHEMBL4811502 0.81 MAOB (0.84) CREBBPNR4A2RAB9AMAOBEP300
SCHEMBL29176621 0.81 MAOB (0.62) CREBBPNR4A2MAOBEP300ALDH1A1
SCHEMBL9163212 0.78 NR4A2 (0.72) NR4A2SRCRAB9ATSHRALDH1A1
SCHEMBL31621504 0.77 NR4A2 (1.00) NR4A2TSHRALDH1A1NPSR1SMN1; SMN2
SCHEMBL1092934 0.77 NR4A2 (1.00) NR4A2TSHRALDH1A1NPSR1SMN1; SMN2
SCHEMBL9165197 0.76 EGFR (0.57) CREBBPNR4A2SRCMAOBEP300
SCHEMBL677770 0.76 RAB9A (1.00) RAB9AALDH1A1SMN1; SMN2TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5464861-A Anticarcinogenic agents WARNER-LAMBERT (US) 1995-11-07 US disclosed
EP-0654024-A1 2-THIOINDOLES (SELENOINDOLES) AND RELATED DISULFIDES (SELENIDES) WHICH INHIBIT PROTEIN TYROSINE KINASES AND WHICH HAVE ANTITUMOR PROPERTIES WARNER-LAMBERT COMPANY (US) 1995-05-24 EP disclosed
WO-1994003427-A1 2-THIOINDOLES (SELENOINDOLES) AND RELATED DISULFIDES (SELENIDES) WHICH INHIBIT PROTEIN TYROSINE KINASES AND WHICH HAVE ANTITUMOR PROPERTIES WARNER-LAMBERT COMPANY (US) 1994-02-17 WO disclosed