SCHEMBL9159683

SCHEMBL9159683

N#Cc1ccc(C(c2ccc(C(F)(F)F)cc2)c2cccnc2)cc1

nearest known ligand 0.78

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 6/20 0.78
CYP3A4 P08684 7/20 0.61
CYP3A5 P20815 3/20 0.61
CFTR P13569 1/20 0.50
SLC6A2 P23975 1/20 0.50
SLC6A4 P31645 1/20 0.50
SLC6A3 Q01959 1/20 0.50
GOPC Q9HD26 1/20 0.50
KIF11 P52732 1/20 0.49
CYP11B2 P19099 2/20 0.45
TRPM8 Q7Z2W7 1/20 0.45
NPC1 O15118 1/20 0.42
HRH3 Q9Y5N1 1/20 0.40
CYP11B1 P15538 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2354875 0.88 CYP19A1 (1.00) CYP19A1CYP3A4CYP3A5CFTRSLC6A2
SCHEMBL9790964 0.88 CYP19A1 (1.00) CYP19A1CYP3A4CYP3A5CFTRSLC6A2
SCHEMBL9790876 0.87 CYP19A1 (0.90) CYP19A1CYP3A4CYP3A5CFTRSLC6A2
Hydrochloric Acid SCHEMBL1507785 0.87 CYP19A1 (0.97) CYP19A1CYP3A4CYP3A5CFTRSLC6A2
SCHEMBL9165271 0.81 CYP19A1 (0.85) CYP19A1CYP3A4CYP3A5CFTRSLC6A2
SCHEMBL5597318 0.76 CYP19A1 (0.74) CYP19A1CYP3A4CYP3A5CFTRSLC6A2
SCHEMBL1507962 0.75 CYP19A1 (0.73) CYP19A1CYP3A4CYP3A5CFTRSLC6A2
SCHEMBL9165268 0.75 CYP19A1 (0.73) CYP19A1CYP3A4CYP3A5CFTRSLC6A2
SCHEMBL1507855 0.74 KIF11 (0.47) CYP19A1CYP3A4CYP3A5KIF11CYP11B2
SCHEMBL10558176 0.73 CYP19A1 (0.71) CYP19A1CYP3A4CYP3A5CFTRSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5473078-A Aromatase inhibiting compounds CIBA-GEIGY CORPORATION (US) 1995-12-05 US disclosed
US-5352795-A Condensing triazolylmethylbenzonitrile with fluorobenzonitrile under basic conditions using alkali metal alkoxide CIBA-GEIGY CORPORATION (US) 1994-10-04 US disclosed
US-5112845-A Inhibitors of estrogen synthesis, veterinary medicine CIBA-GEIGY CORPORATION (US) 1992-05-12 US disclosed
US-4978672-A Alpha-heterocyclc substituted tolunitriles CIBA-GEIGY CORPORATION (US) 1990-12-18 US disclosed