SCHEMBL9164635

SCHEMBL9164635

N#Cc1cccc(C(c2ccccc2)c2nnc[nH]2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 4/20 0.39
GABRB3 P28472 4/20 0.39
GABRA5 P31644 4/20 0.39
GABRA3 P34903 4/20 0.39
GABRA1 P14867 1/20 0.39
IDO1 P14902 2/20 0.38
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
MAOB P27338 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
CYP19A1 P11511 2/20 0.35
TSHR P16473 2/20 0.35
NOTUM Q6P988 1/20 0.35
GRM4 Q14833 1/20 0.34
ALDH1A1 P00352 2/20 0.33
LMNA P02545 1/20 0.33
CRHBP P24387 1/20 0.33
HTT P42858 1/20 0.33
CRHR2 Q13324 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1507964 0.81 CYP19A1 (0.46) HRH3CYP19A1TSHRNOTUM
SCHEMBL9164675 0.75 CYP19A1 (0.68) SLC6A2SLC6A4CYP19A1
SCHEMBL9161325 0.74 CYP19A1 (0.41) IDO1MAOBHRH3CYP19A1TSHR
SCHEMBL9165090 0.73 CYP19A1 (0.38) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL4083138 0.73 ENPP2 (0.47) IDO1SLC6A2SLC6A4CYP19A1TSHR
SCHEMBL9165167 0.72 SLC6A2 (0.40) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL9161362 0.71 CYP19A1 (0.49) MAOBCYP19A1ALDH1A1LMNAHTT
SCHEMBL9159543 0.70 CYP19A1 (0.37) CYP19A1
SCHEMBL9164614 0.70 GUSB (0.37) SLC6A4CYP19A1ALDH1A1
SCHEMBL9167265 0.69 CYP19A1 (0.37) CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5473078-A Aromatase inhibiting compounds CIBA-GEIGY CORPORATION (US) 1995-12-05 US disclosed
US-5352795-A Condensing triazolylmethylbenzonitrile with fluorobenzonitrile under basic conditions using alkali metal alkoxide CIBA-GEIGY CORPORATION (US) 1994-10-04 US disclosed
US-5112845-A Inhibitors of estrogen synthesis, veterinary medicine CIBA-GEIGY CORPORATION (US) 1992-05-12 US disclosed
US-4978672-A Alpha-heterocyclc substituted tolunitriles CIBA-GEIGY CORPORATION (US) 1990-12-18 US disclosed