SCHEMBL9165437

SCHEMBL9165437

O=C(O)C(CO)N1CCNCCNCCN(C(CO)C(=O)O)CC1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.36
OPRD1 P41143 8/20 0.35
SLC6A4 P31645 1/20 0.33
LMNA P02545 1/20 0.33
CHRM5 P08912 1/20 0.33
CHRM3 P20309 1/20 0.33
CA2 P00918 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA9 Q16790 1/20 0.32
OPRM1 P35372 1/20 0.32
CHKA P35790 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30598667 0.98 SIGMAR1 (0.35) SIGMAR1OPRD1SLC6A4LMNACHRM5
SCHEMBL9158636 0.98 SIGMAR1 (0.37) SIGMAR1OPRD1SLC6A4LMNACHRM5
SCHEMBL9161735 0.98 SIGMAR1 (0.37) SIGMAR1OPRD1SLC6A4LMNACHRM5
SCHEMBL9167411 0.96 SIGMAR1 (0.38) SIGMAR1OPRD1SLC6A4LMNACHRM5
SCHEMBL30598663 0.94 SIGMAR1 (0.37) SIGMAR1OPRD1SLC6A4LMNACHRM5
SCHEMBL300399 0.85
SCHEMBL8310688 0.84 SIGMAR1 (0.41) SIGMAR1OPRD1SLC6A4LMNACHRM5
SCHEMBL6423819 0.83 SIGMAR1 (0.41) SIGMAR1OPRD1SLC6A4CHRM5CHRM3
SCHEMBL31492641 0.82 SIGMAR1 (0.39) SIGMAR1OPRD1CHRM5CHRM3CA2
SCHEMBL30914551 0.81 HSD17B10 (0.37) SIGMAR1OPRD1SLC6A4LMNACHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0325762-B1 Macrocyclic chelating agents and chelates thereof BRACCO SPA (IT) 1995-03-22 EP claimed
EP-0325762-A1 Macrocyclic chelating agents and chelates thereof BRACCO S.p.A. (IT) 1989-08-02 EP claimed
EP-0325762-B1 Macrocyclic chelating agents and chelates thereof BRACCO SPA (IT) 1995-03-22 EP disclosed
US-5132409-A Derivatives of 1,4,7,10-Tetraazacyclododecane BRACCO INDUSTRIA CHIMICA S.P.A. (IT) 1992-07-21 US disclosed
EP-0325762-A1 Macrocyclic chelating agents and chelates thereof BRACCO S.p.A. (IT) 1989-08-02 EP disclosed