SCHEMBL9166361

SCHEMBL9166361

Cc1cccc(-n2nc(C(=O)C(C#N)C(=O)Nc3ccccc3)c3c2-c2ccccc2C3)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNA2 P20248 1/20 0.41
CDK2 P24941 1/20 0.41
CCNA1 P78396 1/20 0.41
MAPK13 O15264 1/20 0.40
MAPK12 P53778 1/20 0.40
MAPK11 Q15759 1/20 0.40
MAPK14 Q16539 1/20 0.40
PIK3CD O00329 1/20 0.39
PIK3R2 O00459 1/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CB P42338 1/20 0.39
PIK3CG P48736 1/20 0.39
PIK3R5 Q8WYR1 1/20 0.39
PIK3R3 Q92569 1/20 0.39
TP53 P04637 1/20 0.37
KCNJ6 P48051 3/20 0.36
KCNJ3 P48549 3/20 0.36
KCNJ5 P48544 2/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9173515 0.95 KCNJ6 (0.42) CCNA2CDK2CCNA1PIK3CDPIK3R2
SCHEMBL8135900 0.91 CCNA2 (0.37) CCNA2CDK2CCNA1MAPK13MAPK12
SCHEMBL9174895 0.91 CCNA2 (0.40) CCNA2CDK2CCNA1PIK3CDPIK3R2
SCHEMBL9167950 0.91 RIPK1 (0.37) CCNA2CDK2CCNA1MAPK13MAPK12
SCHEMBL9171530 0.91 RIPK1 (0.41) KCNJ6KCNJ3KCNJ5NPC1RAB9A
SCHEMBL9171526 0.90 MAPK13 (0.41) MAPK13MAPK12MAPK11MAPK14PIK3CD
SCHEMBL9170088 0.90 CCNA2 (0.41) CCNA2CDK2CCNA1PIK3CDPIK3R2
SCHEMBL9176690 0.90 PIK3CD (0.39) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL9176056 0.90 CNR2 (0.40) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL9170069 0.88 PIK3CD (0.41) CCNA2CDK2CCNA1PIK3CDPIK3R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5424308-A Immunomodulating agents FARMITALIA CARLO ERBA S.R.L. (IT) 1995-06-13 US disclosed
EP-0422051-A1 CONDENSED PYRAZOLE 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1991-04-17 EP disclosed
WO-1989012630-A1 CONDENSED PYRAZOLE 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.R.L. (IT) 1989-12-28 WO disclosed
EP-0347773-A1 Condensed Pyrazole 3-oxo-propanenitrile derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1989-12-27 EP disclosed