SCHEMBL9168136

SCHEMBL9168136

CCCCCCCCCCCCCCCCCCOc1cc(N)cc(C(=O)OC)c1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 2/20 0.57
TSHR P16473 2/20 0.50
SMPD1 P17405 3/20 0.49
NPC1 O15118 1/20 0.48
MAPT P10636 1/20 0.48
RAB9A P51151 1/20 0.48
ALDH1A1 P00352 1/20 0.48
TP53 P04637 1/20 0.47
PLA2G4B P0C869 1/20 0.46
BLM P54132 1/20 0.45
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
ESR1 P03372 1/20 0.44
AKR1C4 P17516 1/20 0.44
AKR1C3 P42330 1/20 0.44
AKR1C2 P52895 1/20 0.44
AKR1C1 Q04828 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5095050 0.90 PLA2G2A (0.71) PLA2G2ATSHRSMPD1MAPTTP53
SCHEMBL7089932 0.90 PLA2G2A (0.66) PLA2G2ATSHRSMPD1MAPTTP53
SCHEMBL1568668 0.90 PLA2G2A (0.71) PLA2G2ATSHRSMPD1MAPTTP53
SCHEMBL25327393 0.90 PLA2G2A (0.71) PLA2G2ATSHRSMPD1MAPTTP53
SCHEMBL1822124 0.90 PLA2G2A (0.66) PLA2G2ATSHRSMPD1MAPTTP53
SCHEMBL25328188 0.90 PLA2G2A (0.71) PLA2G2ATSHRSMPD1MAPTTP53
SCHEMBL971768 0.90 PLA2G2A (0.71) PLA2G2ATSHRSMPD1MAPTTP53
SCHEMBL2710788 0.90 PLA2G2A (0.66) PLA2G2ATSHRSMPD1MAPTTP53
SCHEMBL317989 0.90 PLA2G2A (0.71) PLA2G2ATSHRSMPD1MAPTTP53
SCHEMBL5086867 0.90 PLA2G2A (0.71) PLA2G2ATSHRSMPD1MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5446189-A Diester intermediates for diacid enzyme inhibitor HOFFMANN-LA ROCHE INC. (US) 1995-08-29 US disclosed
US-5324747-A Treatment of inflammatory diseases HOFFMANN-LA ROCHE INC. (US) 1994-06-28 US disclosed
EP-0579066-A2 N-substituted anilines F. HOFFMANN-LA ROCHE AG (CH) 1994-01-19 EP disclosed