SCHEMBL9168212

SCHEMBL9168212

CCOC(=O)c1cnc2c(-c3cc(-c4ccccc4)cs3)cnn2c1O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.60
RAB9A P51151 7/20 0.60
SMN1; SMN2 Q16637 7/20 0.60
MAPT P10636 5/20 0.60
NFKB1 P19838 2/20 0.60
NFKB2 Q00653 2/20 0.60
RELA Q04206 2/20 0.60
KDM4E B2RXH2 8/20 0.58
ALDH1A1 P00352 7/20 0.58
HSD17B10 Q99714 4/20 0.58
HPGD P15428 4/20 0.58
TP53 P04637 2/20 0.58
STAT1 P42224 1/20 0.58
LMNA P02545 2/20 0.48
POLB P06746 1/20 0.48
TSHR P16473 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
GAA P10253 2/20 0.46
GPR119 Q8TDV5 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9165628 0.86 SMN1; SMN2 (0.47) NPC1RAB9ASMN1; SMN2MAPTNFKB1
SCHEMBL9165159 0.86 RAB9A (0.42) NPC1RAB9ASMN1; SMN2MAPTNFKB1
SCHEMBL9167744 0.85 KDM4E (0.46) NPC1RAB9ASMN1; SMN2MAPTNFKB1
SCHEMBL9253696 0.85 NPC1 (0.43) NPC1RAB9ASMN1; SMN2MAPTNFKB1
SCHEMBL9249831 0.84 RAB9A (0.40) NPC1RAB9ASMN1; SMN2MAPTNFKB1
SCHEMBL9166610 0.84 MAP2K1 (0.42) NPC1RAB9ASMN1; SMN2MAPTNFKB1
SCHEMBL9172245 0.84 SMN1; SMN2 (0.45) NPC1RAB9ASMN1; SMN2MAPTNFKB1
SCHEMBL9171248 0.84 MAPT (0.60) NPC1RAB9ASMN1; SMN2MAPTNFKB1
SCHEMBL9688778 0.83 NPC1 (0.45) NPC1RAB9ASMN1; SMN2MAPTNFKB1
SCHEMBL9166588 0.83 RAB9A (0.40) NPC1RAB9ASMN1; SMN2MAPTNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5420128-A Pyrimidine derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-05-30 US disclosed
EP-0503099-A1 PYRIMIDINE DERIVATIVE, PRODUCTION THEREOF, AND ANDROGEN INHIBITOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-09-16 EP disclosed