SCHEMBL9170247

SCHEMBL9170247

O=C(O)C(C(=O)O)C1CCCC(=O)C1c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.44
SLC18A3 Q16572 1/20 0.39
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
OPRK1 P41145 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
KDM4E B2RXH2 2/20 0.38
MAPT P10636 3/20 0.36
ALDH1A1 P00352 3/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
HPGD P15428 1/20 0.36
RAB9A P51151 1/20 0.36
CA1 P00915 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
EDNRA P25101 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9171989 0.82 TSHR (0.45) KDM4EL3MBTL1TP53CYP3A4CYP2C9
SCHEMBL23256884 0.78 MCL1 (0.42) MCL1SLC18A3MAPTALDH1A1L3MBTL1
SCHEMBL11484366 0.73 MT-CO2 (0.44) MCL1SLC18A3KMT2AMAPTALDH1A1
SCHEMBL22831008 0.73 SLC6A2 (0.50) KMT2AALDH1A1CYP3A4POLB
SCHEMBL22831009 0.73 SLC6A2 (0.50) KMT2AALDH1A1CYP3A4POLB
SCHEMBL22831007 0.73 SLC6A2 (0.50) KMT2AALDH1A1CYP3A4POLB
SCHEMBL18088734 0.72 CYP3A4 (0.53) KMT2AALDH1A1L3MBTL1NPC1RAB9A
SCHEMBL11475259 0.71 SLC18A3 (0.41) MCL1SLC18A3KMT2AMAPTALDH1A1
SCHEMBL9169697 0.71 SLC18A3 (0.41) SLC18A3PTGS1PTGS2
SCHEMBL8390909 0.68 MEN1 (0.50) MCL1HTTKMT2AALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5387595-A Antiinflammatory agents MERCK & CO., INC. (US) 1995-02-07 US disclosed
WO-1994004487-A1 ALICYCLIC COMPOUNDS AS TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1994-03-03 WO disclosed