SCHEMBL9173573

SCHEMBL9173573

CC(=O)c1cc(C(Cl)Cl)on1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 17/20 0.43
NPC1 O15118 7/20 0.43
RAB9A P51151 7/20 0.43
ALDH1A1 P00352 5/20 0.43
TP53 P04637 3/20 0.43
GAA P10253 1/20 0.43
CYP1A2 P05177 2/20 0.40
CYP2C19 P33261 1/20 0.40
S1PR1 P21453 1/20 0.38
S1PR3 Q99500 1/20 0.38
NFKB1 P19838 1/20 0.37
MAPK1 P28482 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
CYP2D6 P10635 1/20 0.37
MAPT P10636 1/20 0.37
PKM P14618 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1090650 0.81 SMN1; SMN2 (0.55) SMN1; SMN2NPC1RAB9AALDH1A1TP53
SCHEMBL3056764 0.81 SMN1; SMN2 (0.39) SMN1; SMN2NPC1RAB9AALDH1A1TP53
SCHEMBL26523800 0.72 SMN1; SMN2 (0.39) SMN1; SMN2NPC1RAB9AALDH1A1TP53
SCHEMBL13545103 0.71
SCHEMBL1091423 0.71
SCHEMBL26526008 0.71 SMN1; SMN2 (0.36) SMN1; SMN2NPC1RAB9AALDH1A1TP53
SCHEMBL1703668 0.69 ALDH1A1 (0.44) SMN1; SMN2NPC1RAB9AALDH1A1GAA
SCHEMBL31123940 0.68 HCAR2 (0.61) SMN1; SMN2RAB9AALDH1A1GAACYP1A2
SCHEMBL17761981 0.67 MAPT (0.61) SMN1; SMN2NPC1RAB9AALDH1A1TP53
SCHEMBL2328124 0.67 NOTUM (0.43) SMN1; SMN2NPC1RAB9AALDH1A1S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0428340-B1 Heterocyclic compounds ZENECA LTD (GB) 1995-05-31 EP claimed
EP-0428340-A1 Heterocyclic compounds ZENECA LIMITED (GB) 1991-05-22 EP claimed
EP-0428340-B1 Heterocyclic compounds ZENECA LTD (GB) 1995-05-31 EP disclosed
US-5324741-A Heterocyclic isoxazole compounds having nematicidal activity IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-06-28 US disclosed
EP-0428340-A1 Heterocyclic compounds ZENECA LIMITED (GB) 1991-05-22 EP disclosed