SCHEMBL9174168

SCHEMBL9174168

CN1CCC(Sc2c[nH]c3ccccc23)CC1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.52
ATM Q13315 1/20 0.52
HTR6 P50406 6/20 0.47
TUBB4A P04350 1/20 0.44
TUBB P07437 1/20 0.44
TUBA3C P0DPH7 1/20 0.44
TUBA1B P68363 1/20 0.44
TUBA4A P68366 1/20 0.44
TUBB4B P68371 1/20 0.44
TUBB3 Q13509 1/20 0.44
TUBB2A Q13885 1/20 0.44
TUBB8 Q3ZCM7 1/20 0.44
TUBA3E Q6PEY2 1/20 0.44
TUBA1A Q71U36 1/20 0.44
TUBA1C Q9BQE3 1/20 0.44
TUBB6 Q9BUF5 1/20 0.44
TUBB2B Q9BVA1 1/20 0.44
TUBB1 Q9H4B7 1/20 0.44
LMNA P02545 2/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9172692 0.82 HTR1D (0.46) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL9030023 0.81 CYP2C9 (0.62) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL9172798 0.81 SLC6A4 (0.46) ATMHTR6TUBB4ATUBBTUBA3C
SCHEMBL9176587 0.81 IDO1 (0.44) KDM4EATMHTR6TUBB4ATUBB
SCHEMBL9171444 0.81 IDO1 (0.48) HTR6TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL7031652 0.79 HTR2A (0.49) HTR6LMNAHTR1AHTR2ADRD2
SCHEMBL29338311 0.79 CYP1A2 (0.47) KDM4ETUBB4ATUBBTUBA3CTUBA1B
SCHEMBL9173510 0.79 HTR1D (0.49) HTR6HTR1AHTR2APRKCHPRKCD
SCHEMBL9169951 0.79 HTR1A (0.49) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL9031251 0.78 SLC6A4 (0.53) HTR6HTR1ASLC6A4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5418242-A Piperidinylthioindole derivatives, their methods of preparation and pharmaceutical compositions in which they are present, useful especially as analgesics LABORATOIRES UPSA (FR) 1995-05-23 US disclosed
US-5317025-A Piperidinylthioindole derivatives, their methods of preparation and pharmaceutical compositions in which they are present, useful especially as analgesics LABORATOIRES USPA (FR) 1994-05-31 US disclosed