SCHEMBL9177367

SCHEMBL9177367

COC1(C#N)CCN(Cc2ccccc2)C1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.54
CYP3A4 P08684 4/20 0.45
HSD17B10 Q99714 1/20 0.45
SIGMAR1 Q99720 2/20 0.44
CYP2D6 P10635 5/20 0.44
TSHR P16473 3/20 0.44
ALDH1A1 P00352 1/20 0.43
OPRL1 P41146 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22050088 0.91 OPRM1 (0.60) OPRM1CYP3A4HSD17B10SIGMAR1CYP2D6
SCHEMBL28123157 0.86 CYP3A4 (0.45) OPRM1CYP3A4HSD17B10SIGMAR1CYP2D6
SCHEMBL23285142 0.85 OPRM1 (0.50) OPRM1CYP3A4HSD17B10SIGMAR1CYP2D6
SCHEMBL2604321 0.79 OPRM1 (0.56) OPRM1CYP3A4HSD17B10SIGMAR1TSHR
SCHEMBL2275141 0.78 OPRM1 (0.57) OPRM1CYP3A4HSD17B10SIGMAR1CYP2D6
SCHEMBL23089517 0.78 CYP2D6 (0.46) OPRM1CYP3A4SIGMAR1CYP2D6TSHR
SCHEMBL12406526 0.76 CYP3A4 (0.50) CYP3A4HSD17B10SIGMAR1CYP2D6TSHR
SCHEMBL17714545 0.75 OPRM1 (0.51) OPRM1CYP3A4HSD17B10SIGMAR1TSHR
SCHEMBL3893581 0.75 OPRM1 (0.57) OPRM1CYP3A4HSD17B10SIGMAR1CYP2D6
SCHEMBL15325219 0.75 OPRM1 (0.57) OPRM1CYP3A4HSD17B10SIGMAR1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5453422-A Animal growth promoters BAYER AKTIENGESELLSCHAFT (DE) 1995-09-26 US disclosed
US-5284842-A Active against gramnegative bacteria BAYER AKTIENGESELLSCHAFT (DE) 1994-02-08 US disclosed
US-5173484-A Animal growth regulators BAYER AKTIENGESELLSCHAFT (DE) 1992-12-22 US disclosed