SCHEMBL9178666

SCHEMBL9178666

Cc1c(CC(C)(C)C(=O)O)n(Cc2ccc(Cl)cc2)c2ccc(OCc3cccc(-c4ccccc4)n3)cc12

nearest known ligand 0.76

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 13/20 0.76
ALOX5 P09917 7/20 0.67
PTGES2 Q9H7Z7 4/20 0.65
PTGES O14684 1/20 0.64
CYP3A4 P08684 2/20 0.64
CYP2C9 P11712 2/20 0.64
PTGS1 P23219 2/20 0.62
PTGS2 P35354 1/20 0.62
CYP2D6 P10635 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9176433 0.86 ALOX5AP (1.00) ALOX5APALOX5PTGES2PTGESCYP3A4
SCHEMBL2108478 0.86 ALOX5AP (1.00) ALOX5APALOX5CYP3A4CYP2C9PTGS1
SCHEMBL2106671 0.85 ALOX5AP (0.89) ALOX5APALOX5PTGES2CYP3A4CYP2C9
SCHEMBL9584575 0.84 ALOX5AP (0.80) ALOX5APALOX5PTGES2PTGESCYP3A4
SCHEMBL2108140 0.84 ALOX5AP (0.84) ALOX5APALOX5CYP3A4CYP2C9PTGS1
SCHEMBL9044799 0.83 ALOX5AP (0.82) ALOX5APALOX5PTGES2PTGESCYP3A4
SCHEMBL9434427 0.81 ALOX5AP (0.87) ALOX5APALOX5PTGES2PTGESCYP3A4
SCHEMBL9736625 0.81 PTGES2 (0.71) ALOX5APALOX5PTGES2PTGESCYP3A4
SCHEMBL9305688 0.80 ALOX5AP (1.00) ALOX5APALOX5CYP3A4CYP2C9CYP2D6
SCHEMBL2108502 0.80 PTGS1 (0.80) ALOX5APALOX5CYP3A4CYP2C9PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5389650-A Antiinflammatory agents, anticoagulants, antispasmodic agents MERCK FROSST CANADA, INC. (CA) 1995-02-14 US disclosed
EP-0535923-A1 (Azaarylmethoxy)indoles as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA INC. (CA) 1993-04-07 EP disclosed